| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3327064 | 4 | Tmax | = | 4 | hr | ALA3371014 | hr | Rattus norvegicus | |||
| 2. | ALA3327064 | 4 | t1/2 | = | 5.4 | hr | ALA3371013 | hr | Rattus norvegicus | |||
| 3. | ALA3327064 | 4 | Cmax | = | 510 | nM | ALA3371012 | nM | Rattus norvegicus | |||
| 4. | ALA3327064 | 4 | AUC | = | 7304 | nM.hr | ALA3371011 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 5. | ALA3327064 | 4 | t1/2 | = | 36.6 | min | ALA3371010 | hr | Rattus norvegicus | |||
| 6. | ALA3327064 | 4 | IC50 | = | 1.8 | nM | ALA3371009 | 8.74 | nM | Rattus norvegicus | ||
| 7. | ALA3327064 | 4 | Activity | = | 110 | % | ALA3371007 | % | ||||
| 8. | ALA3327064 | 4 | Activity | = | 81.6 | % | ALA3371006 | % | Homo sapiens | |||
| 9. | ALA3327064 | 4 | PPB | = | 85 | % | ALA3371005 | % | Homo sapiens | |||
| 10. | ALA3327064 | 4 | INH | = | 16.5 | % | ALA3371004 | % | Homo sapiens | |||
| 11. | ALA3327064 | 4 | Tmax | = | 4 | hr | ALA3370769 | hr | Mus musculus | |||
| 12. | ALA3327064 | 4 | logP | = | 3.37 | ALA3371019 | ||||||
| 13. | ALA3327064 | 4 | solubility | = | 7.2 | ug ml-1 | ALA3361514 | ug.mL-1 | ||||
| 14. | ALA3327064 | 4 | Ki | = | 0.66 | nM | ALA3361515 | 9.18 | nM | Homo sapiens | ||
| 15. | ALA3327064 | 4 | t1/2 | = | 17.6 | min | ALA3361516 | hr | Homo sapiens | |||
| 16. | ALA3327064 | 4 | AUC | = | 19650 | nM.hr | ALA3370766 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
| 17. | ALA3327064 | 4 | Cmax | = | 1160 | nM | ALA3370767 | nM | Mus musculus | |||
| 18. | ALA3327064 | 4 | t1/2 | = | 6 | hr | ALA3370768 | hr | Mus musculus | |||
| 19. | ALA3327064 | 4 | IC50 | = | 37.5 | nM | ALA3887157 | 7.43 | 312387 | nM | Mus musculus | |
| 20. | ALA3327064 | 4 | IC50 | = | 5.5 | nM | ALA3887156 | 8.26 | 312386 | nM | Mus musculus |
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