| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3327067 | 7 | IC50 | = | 17.8 | nM | ALA3887157 | 7.75 | 312395 | nM | Mus musculus | |
| 2. | ALA3327067 | 7 | IC50 | = | 4 | nM | ALA3887156 | 8.40 | 312394 | nM | Mus musculus | |
| 3. | ALA3327067 | 7 | Activity | 0 | ALA3371017 | Active | Rattus norvegicus | |||||
| 4. | ALA3327067 | 7 | Activity | 0 | ALA3371016 | Dose-dependent effect | Rattus norvegicus | |||||
| 5. | ALA3327067 | 7 | Activity | 0 | ALA3371015 | Active | Rattus norvegicus | |||||
| 6. | ALA3327067 | 7 | Tmax | = | 1 | hr | ALA3371014 | hr | Rattus norvegicus | |||
| 7. | ALA3327067 | 7 | t1/2 | = | 4.9 | hr | ALA3371013 | hr | Rattus norvegicus | |||
| 8. | ALA3327067 | 7 | Cmax | = | 790 | nM | ALA3371012 | nM | Rattus norvegicus | |||
| 9. | ALA3327067 | 7 | AUC | = | 5716 | nM.hr | ALA3371011 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 10. | ALA3327067 | 7 | t1/2 | = | 1.8 | min | ALA3371010 | hr | Rattus norvegicus | |||
| 11. | ALA3327067 | 7 | IC50 | < | 1.25 | nM | ALA3371009 | nM | Rattus norvegicus | |||
| 12. | ALA3327067 | 7 | Activity | = | 107 | % | ALA3371007 | % | ||||
| 13. | ALA3327067 | 7 | Activity | = | 82.6 | % | ALA3371006 | % | Homo sapiens | |||
| 14. | ALA3327067 | 7 | PPB | = | 96.3 | % | ALA3371005 | % | Homo sapiens | |||
| 15. | ALA3327067 | 7 | INH | 0 | ALA3371004 | Not Determined | % | Homo sapiens | ||||
| 16. | ALA3327067 | 7 | Tmax | = | 1 | hr | ALA3370769 | hr | Mus musculus | |||
| 17. | ALA3327067 | 7 | logP | = | 3.84 | ALA3371019 | ||||||
| 18. | ALA3327067 | 7 | solubility | = | 9.2 | ug ml-1 | ALA3361514 | ug.mL-1 | ||||
| 19. | ALA3327067 | 7 | Ki | = | 0.22 | nM | ALA3361515 | 9.66 | nM | Homo sapiens | ||
| 20. | ALA3327067 | 7 | t1/2 | = | 22.3 | min | ALA3361516 | hr | Homo sapiens |
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