| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3327078 | 21 | Tmax | = | 4 | hr | ALA3371014 | hr | Rattus norvegicus | |||
| 2. | ALA3327078 | 21 | t1/2 | = | 4.2 | hr | ALA3371013 | hr | Rattus norvegicus | |||
| 3. | ALA3327078 | 21 | Cmax | = | 297 | nM | ALA3371012 | nM | Rattus norvegicus | |||
| 4. | ALA3327078 | 21 | AUC | = | 2590 | nM.hr | ALA3371011 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 5. | ALA3327078 | 21 | t1/2 | = | 23.7 | min | ALA3371010 | hr | Rattus norvegicus | |||
| 6. | ALA3327078 | 21 | IC50 | = | 20 | nM | ALA3371009 | 7.70 | nM | Rattus norvegicus | ||
| 7. | ALA3327078 | 21 | Activity | = | 108 | % | ALA3371007 | % | ||||
| 8. | ALA3327078 | 21 | Activity | = | 60.6 | % | ALA3371006 | % | Homo sapiens | |||
| 9. | ALA3327078 | 21 | PPB | = | 92.4 | % | ALA3371005 | % | Homo sapiens | |||
| 10. | ALA3327078 | 21 | INH | 0 | ALA3371004 | Not Determined | % | Homo sapiens | ||||
| 11. | ALA3327078 | 21 | Tmax | = | 4 | hr | ALA3370769 | hr | Mus musculus | |||
| 12. | ALA3327078 | 21 | t1/2 | = | 7.7 | hr | ALA3370768 | hr | Mus musculus | |||
| 13. | ALA3327078 | 21 | logP | = | 3.97 | ALA3371019 | ||||||
| 14. | ALA3327078 | 21 | solubility | = | 21.3 | ug ml-1 | ALA3361514 | ug.mL-1 | ||||
| 15. | ALA3327078 | 21 | Ki | = | 0.19 | nM | ALA3361515 | 9.72 | nM | Homo sapiens | ||
| 16. | ALA3327078 | 21 | t1/2 | = | 22.9 | min | ALA3361516 | hr | Homo sapiens | |||
| 17. | ALA3327078 | 21 | AUC | = | 2530 | nM.hr | ALA3370766 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
| 18. | ALA3327078 | 21 | Cmax | = | 195 | nM | ALA3370767 | nM | Mus musculus |
The page will load shortly, Thanks for your patience!