| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3329874 | 28, GK470 | INH | 0 | ALA3365801 | Active | % | Mus musculus | ||||
| 2. | ALA3329874 | 28, GK470 | INH | 0 | ALA3365800 | Active | % | Mus musculus | ||||
| 3. | ALA3329874 | 28, GK470 | INH | 0 | ALA3365798 | Active | % | Mus musculus | ||||
| 4. | ALA3329874 | 28, GK470 | Activity | 0 | ALA3365797 | Non-toxic | Mus musculus | |||||
| 5. | ALA3329874 | 28, GK470 | INH | = | 40 | % | ALA3365795 | % | Homo sapiens | |||
| 6. | ALA3329874 | 28, GK470 | IC50 | = | 0.6 | uM | ALA3365794 | 6.22 | nM | Homo sapiens | ||
| 7. | ALA3329874 | 28, GK470 | INH | > | 90 | % | ALA3365793 | % | Homo sapiens | |||
| 8. | ALA3329874 | 28, GK470 | IC50 | = | 0.3 | uM | ALA3365792 | 6.52 | nM | Homo sapiens | ||
| 9. | ALA3329874 | 28, GK470 | INH | = | 74 | % | ALA3365791 | % | Homo sapiens | |||
| 10. | ALA3329874 | 28, GK470 | INH | = | 41 | % | ALA3365790 | % | ||||
| 11. | ALA3329874 | 28, GK470 | INH | = | 86 | % | ALA3365789 | % | ||||
| 12. | ALA3329874 | 28, GK470 | XI50 | = | 0.011 | mole fraction | ALA3365788 | mole fraction | Homo sapiens | |||
| 13. | ALA3329874 | 28, GK470 | INH | > | 90 | % | ALA3365787 | % | Homo sapiens | |||
| 14. | ALA3329874 | 28, GK470 | AUCt | = | 1861.9 | ng/mL.hr | ALA3362498 | ng.hr.mL-1 | Mus musculus | |||
| 15. | ALA3329874 | 28, GK470 | AUCt | = | 1266.1 | ng/mL.hr | ALA3362497 | ng.hr.mL-1 | Mus musculus | |||
| 16. | ALA3329874 | 28, GK470 | Cmax | = | 2.7 | ug ml-1 | ALA3362496 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Mus musculus | ||
| 17. | ALA3329874 | 28, GK470 | Cmax | = | 234.5 | ng/ml | ALA3362495 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Mus musculus | ||
| 18. | ALA3329874 | 28, GK470 | t1/2 | = | 190 | min | ALA3362494 | hr | Mus musculus | |||
| 19. | ALA3329874 | 28, GK470 | t1/2 | = | 190 | min | ALA3362493 | hr | Homo sapiens | |||
| 20. | ALA3329874 | 28, GK470 | INH | 0 | ALA3362492 | Active | % | Mus musculus |
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