| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3330073 | 9l | IC50 | 0 | ALA3370432 | Not Active | Homo sapiens | |||||
| 2. | ALA3330073 | 9l | IC50 | = | 2.25 | uM | ALA3370431 | 5.65 | nM | Homo sapiens | ||
| 3. | ALA3330073 | 9l | IC50 | = | 55.3 | uM | ALA3370430 | 4.26 | nM | Homo sapiens | ||
| 4. | ALA3330073 | 9l | IC50 | > | 40 | uM | ALA3370429 | nM | Homo sapiens | |||
| 5. | ALA3330073 | 9l | CL(app) | = | 2.01 | L/hr/kg | ALA3370428 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 6. | ALA3330073 | 9l | t1/2 | = | 2.39 | hr | ALA3370427 | hr | Rattus norvegicus | |||
| 7. | ALA3330073 | 9l | MRT | = | 2.71 | hr | ALA3370426 | hr | Rattus norvegicus | |||
| 8. | ALA3330073 | 9l | AUC | = | 4974 | ng/mL.hr | ALA3370425 | ng.hr.mL-1 | Rattus norvegicus | |||
| 9. | ALA3330073 | 9l | AUCt | = | 4467 | ng/mL.hr | ALA3370424 | ng.hr.mL-1 | Rattus norvegicus | |||
| 10. | ALA3330073 | 9l | Cmax | = | 1121 | ng/ml | ALA3370423 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 11. | ALA3330073 | 9l | Tmax | = | 0.5 | hr | ALA3370422 | hr | Rattus norvegicus | |||
| 12. | ALA3330073 | 9l | F | = | 22.8 | % | ALA3370414 | % | Rattus norvegicus | |||
| 13. | ALA3330073 | 9l | t1/2 | = | 2.33 | hr | ALA3370413 | hr | Rattus norvegicus | |||
| 14. | ALA3330073 | 9l | MRT | = | 2.93 | hr | ALA3370412 | hr | Rattus norvegicus | |||
| 15. | ALA3330073 | 9l | AUC | = | 5866 | ng/mL.hr | ALA3370411 | ng.hr.mL-1 | Rattus norvegicus | |||
| 16. | ALA3330073 | 9l | AUCt | = | 5843 | ng/mL.hr | ALA3370181 | ng.hr.mL-1 | Rattus norvegicus | |||
| 17. | ALA3330073 | 9l | Cmax | = | 2711 | ng/ml | ALA3370180 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 18. | ALA3330073 | 9l | Tmax | = | 0.3 | hr | ALA3370178 | hr | Rattus norvegicus | |||
| 19. | ALA3330073 | 9l | Activity | 0 | ALA3370171 | Not Active | Mus musculus | |||||
| 20. | ALA3330073 | 9l | Activity | = | 21.3 | mM | ALA3370170 | mM | Mus musculus |
The page will load shortly, Thanks for your patience!