| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3338090 | 3 | IC50 | = | 3 | nM | ALA3377759 | 8.52 | nM | Homo sapiens | ||
| 2. | ALA3338090 | 3 | IC50 | = | 3 | nM | ALA3377758 | 8.52 | nM | Homo sapiens | ||
| 3. | ALA3338090 | 3 | IC50 | = | 4 | nM | ALA3377757 | 8.40 | nM | Homo sapiens | ||
| 4. | ALA3338090 | 3 | IC50 | = | 4.5 | nM | ALA3377756 | 8.35 | nM | Homo sapiens | ||
| 5. | ALA3338090 | 3 | IC50 | = | 4.9 | nM | ALA3377755 | 8.31 | nM | Homo sapiens | ||
| 6. | ALA3338090 | 3 | IC50 | = | 6.5 | nM | ALA3377754 | 8.19 | nM | Homo sapiens | ||
| 7. | ALA3338090 | 3 | logD | = | 0.9 | ALA3377200 | ||||||
| 8. | ALA3338090 | 3 | solubility | = | 0.87 | mg/ml | ALA3377199 | ug.mL-1 | ||||
| 9. | ALA3338090 | 3 | solubility | = | 0.5 | mg/ml | ALA3377198 | ug.mL-1 | ||||
| 10. | ALA3338090 | 3 | Papp | = | 0.1 | 10'-6 cm/s | ALA3377197 | 10'-6 cm/s | ||||
| 11. | ALA3338090 | 3 | Papp | = | 0.01 | 10'-6 cm/s | ALA3377196 | 10'-6 cm/s | ||||
| 12. | ALA3338090 | 3 | IC50 | = | 10 | nM | ALA3377195 | 8.00 | nM | Homo sapiens | ||
| 13. | ALA3338090 | 3 | pKa | = | 3 | ALA3377194 | ||||||
| 14. | ALA3338090 | 3 | INH | < | 30 | % | ALA3377193 | % | Homo sapiens | |||
| 15. | ALA3338090 | 3 | INH | < | 30 | % | ALA3377192 | % | Homo sapiens | |||
| 16. | ALA3338090 | 3 | t1/2 | = | 2.3 | hr | ALA3377191 | hr | Homo sapiens | |||
| 17. | ALA3338090 | 3 | IC50 | = | 8 | nM | ALA3377190 | 8.10 | nM | Homo sapiens | ||
| 18. | ALA3338090 | 3 | IC50 | = | 5 | nM | ALA3377189 | 8.30 | nM | Homo sapiens | ||
| 19. | ALA3338090 | 3 | IC50 | = | 5 | nM | ALA3778970 | 8.30 | nM | Homo sapiens | ||
| 20. | ALA3338090 | 3 | t1/2 | = | 2.3 | hr | ALA3778972 | hr | Homo sapiens |
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