| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3342554 | 9 | INH | 0 | ALA3387940 | Dose-dependent effect | % | Mus musculus | ||||
| 2. | ALA3342554 | 9 | permeability | > | 4 | % | ALA3387383 | % | Canis lupus familiaris | |||
| 3. | ALA3342554 | 9 | Drug metabolism | < | 20 | % | ALA3387382 | % | Homo sapiens | |||
| 4. | ALA3342554 | 9 | Drug metabolism | < | 20 | % | ALA3387381 | % | Canis lupus familiaris | |||
| 5. | ALA3342554 | 9 | Drug metabolism | < | 20 | % | ALA3387380 | % | Rattus norvegicus | |||
| 6. | ALA3342554 | 9 | Drug metabolism | < | 20 | % | ALA3387379 | % | ||||
| 7. | ALA3342554 | 9 | INH | < | 15 | % | ALA3387378 | % | Homo sapiens | |||
| 8. | ALA3342554 | 9 | INH | < | 15 | % | ALA3387377 | % | Homo sapiens | |||
| 9. | ALA3342554 | 9 | INH | < | 15 | % | ALA3387376 | % | Homo sapiens | |||
| 10. | ALA3342554 | 9 | Vd | < | 1 | L/Kg | ALA3386082 | L.kg-1 | Canis lupus familiaris | |||
| 11. | ALA3342554 | 9 | CL | < | 4 | ml/min.kg | ALA3386081 | mL.min-1.kg-1 | Canis lupus familiaris | |||
| 12. | ALA3342554 | 9 | F | > | 75 | % | ALA3386080 | % | Canis lupus familiaris | |||
| 13. | ALA3342554 | 9 | solubility | = | 1.13 | mg/ml | ALA3386079 | ug.mL-1 | ||||
| 14. | ALA3342554 | 9 | pKa | = | 5 | ALA3386078 | ||||||
| 15. | ALA3342554 | 9 | logD | = | 1.2 | ALA3386077 | ||||||
| 16. | ALA3342554 | 9 | logP | = | 2.24 | ALA3386076 | ||||||
| 17. | ALA3342554 | 9 | INH | 0 | ALA3386074 | Not Active | % | |||||
| 18. | ALA3342554 | 9 | IC50 | = | 3.91 | nM | ALA3385532 | 8.41 | nM | Mus musculus | ||
| 19. | ALA3342554 | 9 | IC50 | = | 12.4 | nM | ALA3385531 | 7.91 | nM | Homo sapiens |
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