| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3342756 | 10 | Activity | 0 | ALA5230046 | Active | Mus musculus | |||||
| 2. | ALA3342756 | 10 | Activity | = | 85.8 | % | ALA5230045 | % | ||||
| 3. | ALA3342756 | 10 | INH | < | 50 | % | ALA5230043 | % | ||||
| 4. | ALA3342756 | 10 | Activity | = | 63.5 | % | ALA5230041 | % | Mus musculus | |||
| 5. | ALA3342756 | 10 | IC50 | = | 16.1 | uM | ALA5230040 | 4.79 | nM | Mus musculus | ||
| 6. | ALA3342756 | 10 | INH | = | 97.4 | % | ALA5230039 | % | Mus musculus | |||
| 7. | ALA3342756 | 10 | Ratio IC50 | = | 2 | ALA4671276 | ||||||
| 8. | ALA3342756 | 10 | Activity | 0 | ALA4671275 | Active | Homo sapiens | |||||
| 9. | ALA3342756 | 10 | IC50 | = | 8.6 | uM | ALA4671274 | 5.07 | nM | |||
| 10. | ALA3342756 | 10 | IC50 | = | 17.7 | uM | ALA4671273 | 4.75 | nM | Homo sapiens | ||
| 11. | ALA3342756 | 10 | IC50 | = | 6.4 | uM | ALA4671272 | 5.19 | nM | Homo sapiens | ||
| 12. | ALA3342756 | 10 | IC50 | = | 6.7 | uM | ALA4671271 | 5.17 | nM | Homo sapiens | ||
| 13. | ALA3342756 | 10 | IC50 | = | 8.4 | uM | ALA4671270 | 5.08 | nM | Homo sapiens | ||
| 14. | ALA3342756 | 10 | Ratio IC50 | = | 1084.3 | ALA3377076 | ||||||
| 15. | ALA3342756 | 10 | IC50 | = | 184.3 | uM | ALA3377075 | nM | Rattus norvegicus | |||
| 16. | ALA3342756 | 10 | IC50 | = | 0.17 | uM | ALA3377074 | 6.77 | nM | Trypanosoma cruzi | ||
| 17. | ALA3342756 | 10 | IC50 | = | 14.3 | uM | ALA3377073 | 4.84 | nM | Trypanosoma brucei rhodesiense | ||
| 18. | ALA3342756 | 10 | IC50 | > | 100 | uM | ALA3377072 | nM | Trypanosoma brucei brucei | |||
| 19. | ALA3342756 | 10 | Selectivity Index | = | 0.7 | ALA3804543 | ||||||
| 20. | ALA3342756 | 10 | IC50 | = | 23.4 | ug ml-1 | ALA3804542 | ug.mL-1 | Homo sapiens |
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