# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3350522 | 1a, n = 6 | Inactivation | > | 90 | % | ALA845789 | % | ||||
2. | ALA3350522 | 1a, n = 6 | Relative affinity | = | 0.28 | ALA839346 | ||||||
3. | ALA3350522 | 1a, n = 6 | Inhibition | = | 33 | % | ALA698381 | % | Rattus norvegicus | |||
4. | ALA3350522 | 1a, n = 6 | Inhibition | = | 35 | % | ALA697558 | % | Rattus norvegicus | |||
5. | ALA3350522 | 1a, n = 6 | Inhibition | = | 23 | % | ALA697397 | % | Rattus norvegicus | |||
6. | ALA3350522 | 1a, n = 6 | Inhibition | = | 23 | % | ALA697736 | % | ||||
7. | ALA3350522 | 1a, n = 6 | Inhibition | = | 0 | % | ALA814472 | % | Homo sapiens | |||
8. | ALA3350522 | 1a, n = 6 | Inhibition | = | 0 | % | ALA814474 | % | Homo sapiens | |||
9. | ALA3350522 | 1a, n = 6 | Loss of inactivation | = | 8 | % | ALA641581 | % | ||||
10. | ALA3350522 | 1a, n = 6 | T1/2 | = | 2 | hr | ALA642806 | hr | Rattus norvegicus | |||
11. | ALA3350522 | 1a, n = 6 | Inactivation | = | 47 | % | ALA640318 | % | ||||
12. | ALA3350522 | 1a, n = 6 | Inactivation | = | 46 | % | ALA640318 | % | ||||
13. | ALA3350522 | 1a, n = 6 | Inactivation | = | 25 | % | ALA640319 | % | ||||
14. | ALA3350522 | 1a, n = 6 | Inactivation | = | 25 | % | ALA640320 | % | ||||
15. | ALA3350522 | 1a, n = 6 | Ki | = | 7.3 | mM | ALA644146 | nM | Rattus norvegicus | |||
16. | ALA3350522 | 1a, n = 6 | Vmax | 0 | ALA632240 | Ability of the 0.43 mM compound to inactivate rat muscle adenylate kinase was determined, after exposing enzyme to 0 mM levels of MgATP | Rattus norvegicus |