# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA109848 | 17 | pKi | = | 6.28 | ALA3056712 | 6.28 | nM | Rattus norvegicus | |||
2. | ALA109848 | 17 | pKi | < | 5 | ALA3056713 | nM | Mesocricetus auratus | ||||
3. | ALA109848 | 17 | pKi | < | 5 | ALA3056710 | nM | Rattus norvegicus | ||||
4. | ALA109848 | 17 | pEC50 | = | 5.89 | ALA3056711 | 5.89 | nM | Oryctolagus cuniculus | |||
5. | ALA109848 | 17 | Efficacy | = | 70 | % | ALA3057222 | % | Oryctolagus cuniculus | |||
6. | ALA109848 | 17 | pEC50 | = | 4.84 | ALA3056709 | 4.84 | nM | Rattus norvegicus | |||
7. | ALA109848 | 17 | Efficacy | = | 35 | % | ALA3057220 | % | Rattus norvegicus | |||
8. | ALA109848 | 17 | Ratio | = | 3.1 | ALA849927 | Canis lupus familiaris | |||||
9. | ALA109848 | 17 | ED delta20 | = | 220 | nM kg-1 | ALA663910 | nM kg-1 | Canis lupus familiaris | |||
10. | ALA109848 | 17 | ED delta5 | = | 68.4 | nM kg-1 | ALA663912 | nM kg-1 | Canis lupus familiaris | |||
11. | ALA109848 | 17 | Selectivity | = | 0.2 | ALA845021 | ||||||
12. | ALA109848 | 17 | Efficacy | = | 100 | % | ALA643882 | % | Rattus norvegicus | |||
13. | ALA109848 | 17 | pD2 | = | 6.64 | ALA645786 | Rattus norvegicus | |||||
14. | ALA109848 | 17 | Selectivity | = | 6 | ALA845022 | ||||||
15. | ALA109848 | 17 | Selectivity | = | 1 | ALA845023 | ||||||
16. | ALA109848 | 17 | Log Ki | = | -5.52 | ALA857772 | 5.52 | nM | Rattus norvegicus | |||
17. | ALA109848 | 17 | Log Ki | = | -6.26 | ALA643232 | 6.26 | nM | Homo sapiens | |||
18. | ALA109848 | 17 | Efficacy | = | 35 | % | ALA647274 | % | Rattus norvegicus | |||
19. | ALA109848 | 17 | pD2 | = | 4.84 | ALA646233 | Rattus norvegicus | |||||
20. | ALA109848 | 17 | Efficacy | = | 70 | % | ALA645471 | % | Oryctolagus cuniculus |