# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA321644 | 11 (+) | pKi | = | 6.6 | ALA3056712 | 6.60 | nM | Rattus norvegicus | |||
2. | ALA321644 | 11 (+) | pKi | < | 5 | ALA3056713 | nM | Mesocricetus auratus | ||||
3. | ALA321644 | 11 (+) | pKi | < | 5 | ALA3056710 | nM | Rattus norvegicus | ||||
4. | ALA321644 | 11 (+) | pEC50 | = | 5.55 | ALA3056711 | 5.55 | nM | Oryctolagus cuniculus | |||
5. | ALA321644 | 11 (+) | Efficacy | = | 64 | % | ALA3057222 | % | Oryctolagus cuniculus | |||
6. | ALA321644 | 11 (+) | pEC50 | 0 | ALA3056709 | Not Active | Rattus norvegicus | |||||
7. | ALA321644 | 11 (+) | pA2 | = | 4.37 | ALA3057214 | 4.37 | nM | Rattus norvegicus | |||
8. | ALA321644 | 11 (+) | pA2 | = | 4.56 | ALA3054763 | 4.56 | nM | Rattus norvegicus | |||
9. | ALA321644 | 11 (+) | Selectivity Index | = | 6.1 | ALA3057217 | Canis lupus familiaris | |||||
10. | ALA321644 | 11 (+) | Ratio | = | 3 | ALA849927 | Canis lupus familiaris | |||||
11. | ALA321644 | 11 (+) | ED delta20 | = | 450 | nM kg-1 | ALA663910 | nM kg-1 | Canis lupus familiaris | |||
12. | ALA321644 | 11 (+) | ED delta5 | = | 0.14 | nM kg-1 | ALA663912 | nM kg-1 | Canis lupus familiaris | |||
13. | ALA321644 | 11 (+) | Selectivity | = | 0.14 | ALA845021 | ||||||
14. | ALA321644 | 11 (+) | Efficacy | = | 100 | % | ALA643882 | % | Rattus norvegicus | |||
15. | ALA321644 | 11 (+) | pD2 | = | 6.59 | ALA645786 | Rattus norvegicus | |||||
16. | ALA321644 | 11 (+) | Selectivity | > | 80 | ALA845022 | ||||||
17. | ALA321644 | 11 (+) | Selectivity | = | 8 | ALA845023 | ||||||
18. | ALA321644 | 11 (+) | Log Ki | < | -5 | ALA857772 | nM | Rattus norvegicus | ||||
19. | ALA321644 | 11 (+) | Log Ki | = | -6.02 | ALA643232 | 6.02 | nM | Homo sapiens | |||
20. | ALA321644 | 11 (+) | pD2 | 0 | ALA646234 | Not Determined | Rattus norvegicus |