# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA111496 | 10 (+) | pKi | = | 7.02 | ALA3056712 | 7.02 | nM | Rattus norvegicus | |||
2. | ALA111496 | 10 (+) | pKi | = | 5.16 | ALA3056713 | 5.16 | nM | Mesocricetus auratus | |||
3. | ALA111496 | 10 (+) | pKi | = | 5.78 | ALA3056710 | 5.78 | nM | Rattus norvegicus | |||
4. | ALA111496 | 10 (+) | pEC50 | = | 6.2 | ALA3056711 | 6.20 | nM | Oryctolagus cuniculus | |||
5. | ALA111496 | 10 (+) | Efficacy | = | 70 | % | ALA3057222 | % | Oryctolagus cuniculus | |||
6. | ALA111496 | 10 (+) | pEC50 | 0 | ALA3056709 | Not Active | Rattus norvegicus | |||||
7. | ALA111496 | 10 (+) | Ratio | = | 3.3 | ALA849927 | Canis lupus familiaris | |||||
8. | ALA111496 | 10 (+) | ED delta20 | = | 34 | nM kg-1 | ALA663910 | nM kg-1 | Canis lupus familiaris | |||
9. | ALA111496 | 10 (+) | ED delta5 | = | 10.5 | nM kg-1 | ALA663912 | nM kg-1 | Canis lupus familiaris | |||
10. | ALA111496 | 10 (+) | Selectivity | = | 7 | ALA845021 | ||||||
11. | ALA111496 | 10 (+) | Efficacy | = | 66 | % | ALA643882 | % | Rattus norvegicus | |||
12. | ALA111496 | 10 (+) | pD2 | = | 5.95 | ALA645786 | Rattus norvegicus | |||||
13. | ALA111496 | 10 (+) | Selectivity | = | 40 | ALA845022 | ||||||
14. | ALA111496 | 10 (+) | Selectivity | = | 3 | ALA845023 | ||||||
15. | ALA111496 | 10 (+) | Log Ki | = | -5.77 | ALA857772 | 5.77 | nM | Rattus norvegicus | |||
16. | ALA111496 | 10 (+) | Log Ki | = | -6.88 | ALA643232 | 6.88 | nM | Homo sapiens | |||
17. | ALA111496 | 10 (+) | pD2 | 0 | ALA646234 | Not Determined | Rattus norvegicus | |||||
18. | ALA111496 | 10 (+) | Efficacy | = | 71 | % | ALA645471 | % | Oryctolagus cuniculus | |||
19. | ALA111496 | 10 (+) | pD2 | = | 6.77 | ALA645473 | Oryctolagus cuniculus | |||||
20. | ALA111496 | 10 (+) | Selectivity | = | 20 | ALA845025 | Rattus norvegicus |