# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3355137 | 17k | INH | = | 50 | % | ALA3387831 | % | ||||
2. | ALA3355137 | 17k | INH | = | 50 | % | ALA3387830 | % | Homo sapiens | |||
3. | ALA3355137 | 17k | INH | = | 50 | % | ALA3387829 | % | Homo sapiens | |||
4. | ALA3355137 | 17k | EC50 | = | 5.5 | uM | ALA3387828 | 5.26 | nM | Homo sapiens | ||
5. | ALA3355137 | 17k | IC50 | = | 6.8 | uM | ALA3387827 | 5.17 | nM | |||
6. | ALA3355137 | 17k | INH | 0 | ALA3387826 | Active | % | Homo sapiens | ||||
7. | ALA3355137 | 17k | INH | 0 | ALA3387825 | Active | % | Homo sapiens | ||||
8. | ALA3355137 | 17k | INH | 0 | ALA3387824 | Active | % | |||||
9. | ALA3355137 | 17k | INH | = | 85 | % | ALA3387816 | % | Mus musculus | |||
10. | ALA3355137 | 17k | fAUC | = | 1020 | ng.hr/ml | ALA3387806 | ng.hr.mL-1 | Mus musculus | |||
11. | ALA3355137 | 17k | fCmax | = | 78 | ng/ml | ALA3387805 | ng/ml | Mus musculus | |||
12. | ALA3355137 | 17k | t1/2 | = | 4.8 | hr | ALA3387804 | hr | Mus musculus | |||
13. | ALA3355137 | 17k | IC50 | = | 0.01 | uM | ALA3387798 | 8.00 | nM | |||
14. | ALA3355137 | 17k | IC50 | = | 0.002 | uM | ALA3387797 | 8.70 | nM | Homo sapiens |