| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3355737 | 4i | INH | = | 70 | % | ALA3390079 | % | Homo sapiens | |||
| 2. | ALA3355737 | 4i | INH | = | 70 | % | ALA3390078 | % | Homo sapiens | |||
| 3. | ALA3355737 | 4i | INH | = | 70 | % | ALA3390077 | % | Homo sapiens | |||
| 4. | ALA3355737 | 4i | Ratio | = | 4.8 | ALA3390076 | Canis lupus familiaris | |||||
| 5. | ALA3355737 | 4i | Papp | = | 12 | 10'-6 cm/s | ALA3390075 | 10'-6 cm/s | Canis lupus familiaris | |||
| 6. | ALA3355737 | 4i | Papp | = | 2.5 | 10'-6 cm/s | ALA3390074 | 10'-6 cm/s | Canis lupus familiaris | |||
| 7. | ALA3355737 | 4i | INH | 0 | ALA3390073 | Not Active | % | Homo sapiens | ||||
| 8. | ALA3355737 | 4i | INH | 0 | ALA3390072 | Not Active | % | Homo sapiens | ||||
| 9. | ALA3355737 | 4i | INH | 0 | ALA3390071 | Not Active | % | Homo sapiens | ||||
| 10. | ALA3355737 | 4i | INH | 0 | ALA3390070 | Not Active | % | Homo sapiens | ||||
| 11. | ALA3355737 | 4i | CLH | = | 16 | ml/min.kg | ALA3390069 | mL.min-1.kg-1 | Homo sapiens | |||
| 12. | ALA3355737 | 4i | Kinetic_solubility | <= | 1 | uM | ALA3390068 | nM | ||||
| 13. | ALA3355737 | 4i | IC50 | = | 180 | nM | ALA3390067 | 6.75 | nM | Homo sapiens | ||
| 14. | ALA3355737 | 4i | Selectivity ratio | = | 182 | ALA3390066 | ||||||
| 15. | ALA3355737 | 4i | Ki | = | 0.17 | nM | ALA3389531 | 9.77 | nM | Homo sapiens |
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