Activities

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Activities

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#	Name	Compound Key	Action Type	Relation	Activity Value	Units	Assay ID	Assay Description	Assay	Assay Organism
1.	ALA3360855	EPZ, EPZ005687	F	=	47	%	ALA3772962		%	Mus musculus
2.	ALA3360855	EPZ, EPZ005687	Vdss	=	0.49	L/Kg	ALA3772961		L.kg-1	Mus musculus
3.	ALA3360855	EPZ, EPZ005687	AUC	=	2900	hr.ng/ml	ALA3772960		ng.hr.mL-1	Mus musculus
4.	ALA3360855	EPZ, EPZ005687	CL	=	11	ml/min.kg	ALA3772959		mL.min-1.kg-1	Mus musculus
5.	ALA3360855	EPZ, EPZ005687	EC50	=	2.9	uM	ALA3772958	5.54	nM	Homo sapiens
6.	ALA3360855	EPZ, EPZ005687	IC50	=	54	nM	ALA5138242	7.27	nM	Homo sapiens
7.	ALA3360855	EPZ, EPZ005687	IC50	=	2.9	uM	ALA5123928	5.54	nM	Homo sapiens
8.	ALA3360855	EPZ, EPZ005687	Ki	=	24	nM	ALA5123927	7.62	nM
9.	ALA3360855	EPZ, EPZ005687	IC50	=	54	nM	ALA5123926	7.27	nM	Homo sapiens
10.	ALA3360855	EPZ, EPZ005687	Selectivity ratio	>	500		ALA3421449
11.	ALA3360855	EPZ, EPZ005687	IC50	=	80	nM	ALA3417982	7.10	nM	Homo sapiens
12.	ALA3360855	EPZ, EPZ005687	Selectivity ratio	=	5		ALA3417981
13.	ALA3360855	EPZ, EPZ005687	Selectivity ratio	=	50		ALA3421461
14.	ALA3360855	EPZ, EPZ005687	Selectivity ratio	>	500		ALA3421460
15.	ALA3360855	EPZ, EPZ005687	Selectivity ratio	>	500		ALA3421459
16.	ALA3360855	EPZ, EPZ005687	Selectivity ratio	>	500		ALA3421458
17.	ALA3360855	EPZ, EPZ005687	Selectivity ratio	>	500		ALA3421457
18.	ALA3360855	EPZ, EPZ005687	Selectivity ratio	>	500		ALA3421456
19.	ALA3360855	EPZ, EPZ005687	Selectivity ratio	>	500		ALA3421455
20.	ALA3360855	EPZ, EPZ005687	Selectivity ratio	>	500		ALA3421454