# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3360967 | 8 | Efficacy | = | 95 | % | ALA3378884 | % | Homo sapiens | |||
2. | ALA3360967 | 8 | Efficacy | = | 66 | % | ALA3377016 | % | Homo sapiens | |||
3. | ALA3360967 | 8 | Drug uptake | = | 1 | uM | ALA3377022 | uM | Mus musculus | |||
4. | ALA3360967 | 8 | Cp | = | 0.3 | uM | ALA3377021 | uM | Mus musculus | |||
5. | ALA3360967 | 8 | Cp | = | 6.6 | uM | ALA3377020 | uM | Mus musculus | |||
6. | ALA3360967 | 8 | Efficacy | = | 65 | % | ALA3377018 | % | Homo sapiens | |||
7. | ALA3360967 | 8 | Ki | = | 300 | nM | ALA3377012 | 6.52 | nM | Homo sapiens | ||
8. | ALA3360967 | 8 | Ki | = | 31 | nM | ALA3377013 | 7.51 | nM | Homo sapiens | ||
9. | ALA3360967 | 8 | EC50 | = | 320 | nM | ALA3377014 | 6.50 | nM | Homo sapiens | ||
10. | ALA3360967 | 8 | EC50 | = | 230 | nM | ALA3377015 | 6.64 | nM | Homo sapiens | ||
11. | ALA3360967 | 8 | EC50 | = | 38 | nM | ALA3377017 | 7.42 | nM | Homo sapiens |