# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3360971 | 14 | Efficacy | = | 31 | % | ALA3378885 | % | Homo sapiens | |||
2. | ALA3360971 | 14 | Efficacy | = | 32 | % | ALA3378884 | % | Homo sapiens | |||
3. | ALA3360971 | 14 | Drug uptake | = | 13.2 | uM | ALA3377022 | uM | Mus musculus | |||
4. | ALA3360971 | 14 | Cp | = | 2 | uM | ALA3377021 | uM | Mus musculus | |||
5. | ALA3360971 | 14 | Cp | = | 14 | uM | ALA3377020 | uM | Mus musculus | |||
6. | ALA3360971 | 14 | EC50 | = | 8.3 | nM | ALA3377019 | 8.08 | nM | Homo sapiens | ||
7. | ALA3360971 | 14 | Efficacy | = | 31 | % | ALA3377018 | % | Homo sapiens | |||
8. | ALA3360971 | 14 | EC50 | = | 140 | nM | ALA3377017 | 6.85 | nM | Homo sapiens | ||
9. | ALA3360971 | 14 | Ki | = | 1600 | nM | ALA3377012 | 5.80 | nM | Homo sapiens | ||
10. | ALA3360971 | 14 | Ki | = | 59 | nM | ALA3377013 | 7.23 | nM | Homo sapiens | ||
11. | ALA3360971 | 14 | EC50 | > | 10000 | nM | ALA3377014 | nM | Homo sapiens | |||
12. | ALA3360971 | 14 | EC50 | = | 600 | nM | ALA3377015 | 6.22 | nM | Homo sapiens |