# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3394848 | PE-8 | Selectivity Index | = | 434 | ALA3395539 | ||||||
2. | ALA3394848 | PE-8 | Ki | = | 521 | nM | ALA3395398 | 6.28 | nM | Homo sapiens | ||
3. | ALA3394848 | PE-8 | Ki | = | 1.3 | nM | ALA3395399 | 8.89 | nM | Homo sapiens | ||
4. | ALA3394848 | PE-8 | INH | = | 6.7 | uM | ALA3868328 | uM | Homo sapiens | |||
5. | ALA3394848 | PE-8 | INH | = | 3.8 | uM | ALA3868329 | uM | Homo sapiens | |||
6. | ALA3394848 | PE-8 | PPB | > | 99 | % | ALA3868336 | % | ||||
7. | ALA3394848 | PE-8 | PPB | > | 99 | % | ALA3868347 | % | ||||
8. | ALA3394848 | PE-8 | solubility | < | 26 | uM | ALA3868346 | nM | ||||
9. | ALA3394848 | PE-8 | solubility | < | 26 | uM | ALA3868345 | nM | ||||
10. | ALA3394848 | PE-8 | IC50 | = | 1307 | nM | ALA3868324 | 5.88 | nM | Rattus norvegicus | ||
11. | ALA3394848 | PE-8 | IC50 | = | 11 | nM | ALA3868337 | 7.96 | nM | Rattus norvegicus | ||
12. | ALA3394848 | PE-8 | Ratio IC50 | = | 119 | ALA3868344 | ||||||
13. | ALA3394848 | PE-8 | IC50 | = | 4184 | nM | ALA3868342 | 5.38 | nM | Homo sapiens | ||
14. | ALA3394848 | PE-8 | IC50 | = | 89 | nM | ALA3868341 | 7.05 | nM | |||
15. | ALA3394848 | PE-8 | Ratio IC50 | = | 47 | ALA3868343 | ||||||
16. | ALA3394848 | PE-8 | Ratio Ki | = | 400 | ALA3868340 | ||||||
17. | ALA3394848 | PE-8 | Ki | = | 521 | nM | ALA3868339 | 6.28 | nM | Homo sapiens | ||
18. | ALA3394848 | PE-8 | Ki | = | 1.3 | nM | ALA3868338 | 8.89 | nM |