# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3398236 | (R)-21n | t1/2 | = | 2 | hr | ALA3398871 | hr | Rattus norvegicus | |||
2. | ALA3398236 | (R)-21n | F | = | 76 | % | ALA3398870 | % | Rattus norvegicus | |||
3. | ALA3398236 | (R)-21n | EC50 | = | 140 | nM | ALA3398868 | 6.85 | nM | Homo sapiens | ||
4. | ALA3398236 | (R)-21n | Activity | 0 | ALA3398865 | Not Active | Rattus norvegicus | |||||
5. | ALA3398236 | (R)-21n | Activity | 0 | ALA3398864 | Not Active | Rattus norvegicus | |||||
6. | ALA3398236 | (R)-21n | IC50 | = | 62 | nM | ALA3399051 | 7.21 | nM | Homo sapiens | ||
7. | ALA3398236 | (R)-21n | EC50 | = | 48 | nM | ALA3399050 | 7.32 | nM | Homo sapiens | ||
8. | ALA3398236 | (R)-21n | Intrinsic activity | = | 100 | % | ALA3399049 | % | Rattus norvegicus | |||
9. | ALA3398236 | (R)-21n | EC50 | = | 200 | nM | ALA3399048 | 6.70 | nM | Rattus norvegicus | ||
10. | ALA3398236 | (R)-21n | Intrinsic activity | = | 98 | % | ALA3399047 | % | Homo sapiens | |||
11. | ALA3398236 | (R)-21n | EC50 | = | 6 | nM | ALA3399046 | 8.22 | nM | Homo sapiens |