# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3398292 | 6, mixture of stereoisomers | Ratio IC50 | = | 3.7 | ALA3399095 | Homo sapiens | |||||
2. | ALA3398292 | 6, mixture of stereoisomers | IC50 | = | 34 | umol/L | ALA3399094 | 4.47 | nM | Homo sapiens | ||
3. | ALA3398292 | 6, mixture of stereoisomers | IC50 | = | 9.2 | umol/L | ALA3399093 | 5.04 | nM | Homo sapiens | ||
4. | ALA3398292 | 6, mixture of stereoisomers | Kcat/Km | = | 2 | 10'6/M/s | ALA3399092 | 10'6/M/s | Homo sapiens | |||
5. | ALA3398292 | 6, mixture of stereoisomers | Ratio IC50 | = | 2.5 | ALA4009129 | ||||||
6. | ALA3398292 | 6, mixture of stereoisomers | IC50 | = | 30 | uM | ALA4009128 | 4.52 | nM | Homo sapiens | ||
7. | ALA3398292 | 6, mixture of stereoisomers | IC50 | = | 12 | uM | ALA4009139 | 4.92 | nM | Homo sapiens | ||
8. | ALA3398292 | 6, mixture of stereoisomers | Activity | = | -1.09 | V | ALA4009138 | V | ||||
9. | ALA3398292 | 6, mixture of stereoisomers | Selectivity ratio | = | 1.59 | ALA4009137 | ||||||
10. | ALA3398292 | 6, mixture of stereoisomers | Activity | = | 782 | micromol/min | ALA4009136 | micromol/min | Homo sapiens | |||
11. | ALA3398292 | 6, mixture of stereoisomers | Activity | = | 1247 | micromol/min | ALA4009135 | micromol/min | Homo sapiens | |||
12. | ALA3398292 | 6, mixture of stereoisomers | Activity | = | 100 | % | ALA5113941 | % | Plasmodium berghei | |||
13. | ALA3398292 | 6, mixture of stereoisomers | IC50 | = | 0.845 | uM | ALA5113940 | 6.07 | nM | Plasmodium falciparum |