# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3398294 | 8, mixture of stereoisomers | Ratio IC50 | = | 4.9 | ALA3399095 | Homo sapiens | |||||
2. | ALA3398294 | 8, mixture of stereoisomers | IC50 | = | 79 | umol/L | ALA3399094 | 4.10 | nM | Homo sapiens | ||
3. | ALA3398294 | 8, mixture of stereoisomers | IC50 | = | 16 | umol/L | ALA3399093 | 4.80 | nM | Homo sapiens | ||
4. | ALA3398294 | 8, mixture of stereoisomers | Kcat/Km | = | 2.4 | 10'6/M/s | ALA3399092 | 10'6/M/s | Homo sapiens | |||
5. | ALA3398294 | 8, mixture of stereoisomers | Activity | = | 1380 | micromol/min | ALA3399096 | micromol/min | Homo sapiens | |||
6. | ALA3398294 | 8, mixture of stereoisomers | Ratio IC50 | = | 1.73 | ALA4009129 | ||||||
7. | ALA3398294 | 8, mixture of stereoisomers | IC50 | = | 19 | uM | ALA4009128 | 4.72 | nM | Homo sapiens | ||
8. | ALA3398294 | 8, mixture of stereoisomers | IC50 | = | 11 | uM | ALA4009139 | 4.96 | nM | Homo sapiens | ||
9. | ALA3398294 | 8, mixture of stereoisomers | Activity | = | -1.1 | V | ALA4009138 | V | ||||
10. | ALA3398294 | 8, mixture of stereoisomers | Selectivity ratio | = | 1.7 | ALA4009137 | ||||||
11. | ALA3398294 | 8, mixture of stereoisomers | Activity | = | 764 | micromol/min | ALA4009136 | micromol/min | Homo sapiens | |||
12. | ALA3398294 | 8, mixture of stereoisomers | Activity | = | 1300 | micromol/min | ALA4009135 | micromol/min | Homo sapiens | |||
13. | ALA3398294 | 8, mixture of stereoisomers | Activity | = | 80 | % | ALA5113941 | % | Plasmodium berghei | |||
14. | ALA3398294 | 8, mixture of stereoisomers | IC50 | = | 0.63 | uM | ALA5113940 | 6.20 | nM | Plasmodium falciparum |