# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3408015 | 54 | Activity | = | 45 | % | ALA4384328 | % | Mus musculus | |||
2. | ALA3408015 | 54 | IC50 | = | 0.4 | uM | ALA4384327 | 6.40 | nM | |||
3. | ALA3408015 | 54 | IC50 | = | 3.9 | uM | ALA4384350 | 5.41 | nM | |||
4. | ALA3408015 | 54 | IC50 | = | 3.1 | uM | ALA4384349 | 5.51 | nM | |||
5. | ALA3408015 | 54 | Activity | = | 1.2 | % | ALA4384347 | % | ||||
6. | ALA3408015 | 54 | Activity | = | 8.1 | % | ALA4384345 | % | ||||
7. | ALA3408015 | 54 | INH | 0 | ALA4384343 | Not Active | % | |||||
8. | ALA3408015 | 54 | INH | 0 | ALA4384341 | Not Active | % | |||||
9. | ALA3408015 | 54 | Kinetic_solubility | = | 2.6 | 10'-6mg/ml | ALA4384339 | ug.mL-1 | ||||
10. | ALA3408015 | 54 | Kinetic_solubility | = | 6.2 | 10'-7mg/ml | ALA4384338 | ug.mL-1 | ||||
11. | ALA3408015 | 54 | CLH | = | 12 | ml/min | ALA4384337 | ml/min | ||||
12. | ALA3408015 | 54 | t1/2 | = | 57 | min | ALA4384336 | hr | ||||
13. | ALA3408015 | 54 | INH | 0 | ALA3413041 | Dose-dependent effect | % | |||||
14. | ALA3408015 | 54 | K | > | 100 | uM | ALA3413044 | uM | Homo sapiens | |||
15. | ALA3408015 | 54 | Activity | = | 2.7 | % | ALA3413043 | % | Mus musculus | |||
16. | ALA3408015 | 54 | INH | = | 0.67 | % | ALA3413041 | % | ||||
17. | ALA3408015 | 54 | IC50 | = | 0.4 | uM | ALA3413040 | 6.40 | nM | |||
18. | ALA3408015 | 54 | INH | 0 | ALA3413040 | Dose-dependent effect | % | |||||
19. | ALA3408015 | 54 | INH | = | 0.7 | % | ALA3413038 | % | ||||
20. | ALA3408015 | 54 | INH | = | 45.3 | % | ALA3413039 | % | Mus musculus |