# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3408158 | 59 | INH | 0 | ALA3413041 | Dose-dependent effect | % | |||||
2. | ALA3408158 | 59 | K | > | 100 | uM | ALA3413044 | uM | Homo sapiens | |||
3. | ALA3408158 | 59 | Activity | = | 1.8 | % | ALA3413043 | % | Mus musculus | |||
4. | ALA3408158 | 59 | INH | = | 1.8 | % | ALA3413041 | % | ||||
5. | ALA3408158 | 59 | IC50 | = | 0.98 | uM | ALA3413040 | 6.01 | nM | |||
6. | ALA3408158 | 59 | INH | 0 | ALA3413040 | Dose-dependent effect | % | |||||
7. | ALA3408158 | 59 | INH | = | 2.5 | % | ALA3413038 | % | ||||
8. | ALA3408158 | 59 | INH | = | 7 | % | ALA3413039 | % | Mus musculus | |||
9. | ALA3408158 | 59 | Kinetic_solubility | = | 6.8 | 10'-4mg/ml | ALA4384339 | 10'-4mg/ml | ||||
10. | ALA3408158 | 59 | Kinetic_solubility | = | 2.7 | 10'-4mg/ml | ALA4384338 | 10'-4mg/ml | ||||
11. | ALA3408158 | 59 | CLH | < | 3 | ml/min | ALA4384337 | ml/min | ||||
12. | ALA3408158 | 59 | t1/2 | > | 231 | min | ALA4384336 | hr |