# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3410048 | 18n | IC50 | = | 53 | uM | ALA5244624 | nM | Homo sapiens | |||
2. | ALA3410048 | 18n | F | = | 24 | % | ALA3411324 | % | Rattus norvegicus | |||
3. | ALA3410048 | 18n | Cmax | = | 10.6 | uM | ALA3411323 | nM | Rattus norvegicus | |||
4. | ALA3410048 | 18n | AUC | = | 19.4 | uM.hr | ALA3411322 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
5. | ALA3410048 | 18n | t1/2 | = | 2.2 | hr | ALA3411321 | hr | Rattus norvegicus | |||
6. | ALA3410048 | 18n | Vd | = | 0.3 | L/Kg | ALA3411320 | L.kg-1 | Rattus norvegicus | |||
7. | ALA3410048 | 18n | CL | = | 2.1 | ml/min.kg | ALA3411319 | mL.min-1.kg-1 | Rattus norvegicus | |||
8. | ALA3410048 | 18n | IC50 | = | 730 | nM | ALA3411315 | 6.14 | nM | Rattus norvegicus | ||
9. | ALA3410048 | 18n | t1/2 | = | 40 | min | ALA3411314 | hr | Rattus norvegicus | |||
10. | ALA3410048 | 18n | t1/2 | = | 56 | min | ALA3411313 | hr | Homo sapiens | |||
11. | ALA3410048 | 18n | INH | = | 2 | % | ALA3411306 | % | Homo sapiens | |||
12. | ALA3410048 | 18n | INH | = | -4 | % | ALA3411305 | % | Homo sapiens | |||
13. | ALA3410048 | 18n | INH | = | 8 | % | ALA3411304 | % | Homo sapiens | |||
14. | ALA3410048 | 18n | INH | = | -8 | % | ALA3411303 | % | Homo sapiens | |||
15. | ALA3410048 | 18n | IC50 | > | 10000 | nM | ALA3411302 | nM | Homo sapiens | |||
16. | ALA3410048 | 18n | IC50 | > | 20000 | nM | ALA3411301 | nM | Homo sapiens | |||
17. | ALA3410048 | 18n | IC50 | > | 10000 | nM | ALA3411299 | nM | Homo sapiens | |||
18. | ALA3410048 | 18n | IC50 | = | 53 | nM | ALA3411298 | 7.28 | nM | Homo sapiens |