| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3415342 | (+/-)-21w | INH | > | 95 | % | ALA3418720 | % | Homo sapiens | |||
| 2. | ALA3415342 | (+/-)-21w | INH | 0 | ALA3418723 | Dose-dependent effect | % | Mus musculus | ||||
| 3. | ALA3415342 | (+/-)-21w | INH | 0 | ALA3420660 | Active | % | Homo sapiens | ||||
| 4. | ALA3415342 | (+/-)-21w | beta t1/2 | = | 77.2 | min | ALA3420659 | hr | Rattus norvegicus | |||
| 5. | ALA3415342 | (+/-)-21w | AUClast | = | 212 | microg.min/mL | ALA3420658 | ng.hr.mL-1 | Rattus norvegicus | |||
| 6. | ALA3415342 | (+/-)-21w | F | = | 86 | % | ALA3420657 | % | Rattus norvegicus | |||
| 7. | ALA3415342 | (+/-)-21w | t1/2 | = | 129 | min | ALA3420656 | hr | Rattus norvegicus | |||
| 8. | ALA3415342 | (+/-)-21w | Cmax | = | 400 | ng/ml | ALA3420655 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 9. | ALA3415342 | (+/-)-21w | AUClast | = | 91 | microg.min/mL | ALA3420654 | ng.hr.mL-1 | Rattus norvegicus | |||
| 10. | ALA3415342 | (+/-)-21w | Activity | 0 | ALA3420653 | Active | Mus musculus | |||||
| 11. | ALA3415342 | (+/-)-21w | Activity | 0 | ALA3420652 | Active | Mus musculus | |||||
| 12. | ALA3415342 | (+/-)-21w | Activity | 0 | ALA3420650 | Active | Mus musculus | |||||
| 13. | ALA3415342 | (+/-)-21w | Activity | 0 | ALA3420651 | Active | Mus musculus | |||||
| 14. | ALA3415342 | (+/-)-21w | Activity | 0 | ALA3420649 | Active | Mus musculus | |||||
| 15. | ALA3415342 | (+/-)-21w | Activity | 0 | ALA3420648 | Active | Mus musculus | |||||
| 16. | ALA3415342 | (+/-)-21w | Activity | 0 | ALA3418725 | Active | Rattus norvegicus | |||||
| 17. | ALA3415342 | (+/-)-21w | INH | = | 76 | % | ALA3418724 | % | Rattus norvegicus | |||
| 18. | ALA3415342 | (+/-)-21w | IC50 | > | 60 | uM | ALA3418723 | nM | Mus musculus | |||
| 19. | ALA3415342 | (+/-)-21w | INH | = | 5.05 | % | ALA3418722 | % | Homo sapiens | |||
| 20. | ALA3415342 | (+/-)-21w | INH | = | 16 | % | ALA3418721 | % | Mus musculus |
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