# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3426030 | 78b | Retention_time | = | 1.16 | min | ALA3429030 | min | ||||
2. | ALA3426030 | 78b | AUC/dose | = | 371 | ng/hr/ml | ALA3428894 | ng/hr/ml | Mus musculus | |||
3. | ALA3426030 | 78b | Cmax | = | 1110 | ng/ml | ALA3428890 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Mus musculus | ||
4. | ALA3426030 | 78b | beta t1/2 | = | 1.6 | hr | ALA3428370 | hr | Mus musculus | |||
5. | ALA3426030 | 78b | Vdss | = | 1.2 | L/Kg | ALA3428366 | L.kg-1 | Mus musculus | |||
6. | ALA3426030 | 78b | CL | = | 44.7 | ml/min.kg | ALA3428364 | mL.min-1.kg-1 | Mus musculus | |||
7. | ALA3426030 | 78b | solubility | = | 350 | uM | ALA3428363 | nM | ||||
8. | ALA3426030 | 78b | permeability | = | 200 | nm/s | ALA3428362 | nm/s | Canis lupus familiaris | |||
9. | ALA3426030 | 78b | Ki | = | 14 | nM | ALA3428361 | 7.85 | nM | Homo sapiens | ||
10. | ALA3426030 | 78b | IC50 | = | 15 | nM | ALA3428360 | 7.82 | nM | Mus musculus | ||
11. | ALA3426030 | 78b | IC50 | = | 89 | nM | ALA3428359 | 7.05 | nM | Homo sapiens |