| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3426035 | 79c | Retention_time | = | 1.45 | min | ALA3429030 | min | ||||
| 2. | ALA3426035 | 79c | AUC/dose | = | 2030 | ng/hr/ml | ALA3428894 | ng/hr/ml | Mus musculus | |||
| 3. | ALA3426035 | 79c | AUC/dose | = | 930 | ng/hr/ml | ALA3428893 | ng/hr/ml | Mus musculus | |||
| 4. | ALA3426035 | 79c | Cmax | = | 2500 | ng/ml | ALA3428890 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Mus musculus | ||
| 5. | ALA3426035 | 79c | Cmax | = | 3810 | ng/ml | ALA3428375 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Mus musculus | ||
| 6. | ALA3426035 | 79c | F | = | 46 | % | ALA3428373 | % | Mus musculus | |||
| 7. | ALA3426035 | 79c | beta t1/2 | = | 0.46 | hr | ALA3428370 | hr | Mus musculus | |||
| 8. | ALA3426035 | 79c | beta t1/2 | = | 1.3 | hr | ALA3428369 | hr | Mus musculus | |||
| 9. | ALA3426035 | 79c | Vdss | = | 0.32 | L/Kg | ALA3428366 | L.kg-1 | Mus musculus | |||
| 10. | ALA3426035 | 79c | CL | = | 8.9 | ml/min.kg | ALA3428364 | mL.min-1.kg-1 | Mus musculus | |||
| 11. | ALA3426035 | 79c | solubility | >= | 323 | uM | ALA3428363 | nM | ||||
| 12. | ALA3426035 | 79c | permeability | = | 195 | nm/s | ALA3428362 | nm/s | Canis lupus familiaris | |||
| 13. | ALA3426035 | 79c | Ki | = | 0.7 | nM | ALA3428361 | 9.15 | nM | Homo sapiens | ||
| 14. | ALA3426035 | 79c | IC50 | = | 1.6 | nM | ALA3428360 | 8.80 | nM | Mus musculus | ||
| 15. | ALA3426035 | 79c | IC50 | = | 10 | nM | ALA3428359 | 8.00 | nM | Homo sapiens |
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