| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3426039 | 79d | Retention_time | = | 1.44 | min | ALA3429030 | min | ||||
| 2. | ALA3426039 | 79d | AUC/dose | = | 497 | ng/hr/ml | ALA3428895 | ng/hr/ml | Mus musculus | |||
| 3. | ALA3426039 | 79d | AUC/dose | = | 443 | ng/hr/ml | ALA3428892 | ng/hr/ml | Mus musculus | |||
| 4. | ALA3426039 | 79d | Cmax | = | 1480 | ng/ml | ALA3428891 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Mus musculus | ||
| 5. | ALA3426039 | 79d | Cmax | = | 6250 | ng/ml | ALA3428374 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Mus musculus | ||
| 6. | ALA3426039 | 79d | F | = | 89 | % | ALA3428372 | % | Mus musculus | |||
| 7. | ALA3426039 | 79d | beta t1/2 | = | 1.2 | hr | ALA3428371 | hr | Mus musculus | |||
| 8. | ALA3426039 | 79d | beta t1/2 | = | 3.2 | hr | ALA3428368 | hr | Mus musculus | |||
| 9. | ALA3426039 | 79d | Vdss | = | 1.1 | L/Kg | ALA3428367 | L.kg-1 | Mus musculus | |||
| 10. | ALA3426039 | 79d | CL | = | 33.4 | ml/min.kg | ALA3428365 | mL.min-1.kg-1 | Mus musculus | |||
| 11. | ALA3426039 | 79d | solubility | >= | 340 | uM | ALA3428363 | nM | ||||
| 12. | ALA3426039 | 79d | permeability | = | 300 | nm/s | ALA3428362 | nm/s | Canis lupus familiaris | |||
| 13. | ALA3426039 | 79d | Ki | = | 0.45 | nM | ALA3428361 | 9.35 | nM | Homo sapiens | ||
| 14. | ALA3426039 | 79d | IC50 | = | 1.4 | nM | ALA3428360 | 8.85 | nM | Mus musculus | ||
| 15. | ALA3426039 | 79d | IC50 | = | 15 | nM | ALA3428359 | 7.82 | nM | Homo sapiens |
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