# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3426891 | (R)-9b | IC50 | = | 56 | nM | ALA3429155 | 7.25 | nM | Homo sapiens | ||
2. | ALA3426891 | (R)-9b | solubility | = | 1 | mg/ml | ALA3429154 | ug.mL-1 | ||||
3. | ALA3426891 | (R)-9b | t1/2 | > | 6 | hr | ALA3429153 | hr | Homo sapiens | |||
4. | ALA3426891 | (R)-9b | IC50 | = | 438 | nM | ALA3429152 | 6.36 | nM | Homo sapiens | ||
5. | ALA3426891 | (R)-9b | IC50 | = | 124 | nM | ALA3429151 | 6.91 | nM | Homo sapiens | ||
6. | ALA3426891 | (R)-9b | IC50 | = | 136 | nM | ALA3429150 | 6.87 | nM | Homo sapiens | ||
7. | ALA3426891 | (R)-9b | IC50 | = | 143 | nM | ALA3429149 | 6.84 | nM | Homo sapiens | ||
8. | ALA3426891 | (R)-9b | IC50 | = | 154 | nM | ALA3429148 | 6.81 | nM | Homo sapiens | ||
9. | ALA3426891 | (R)-9b | IC50 | = | 206 | nM | ALA3429147 | 6.69 | nM | Homo sapiens | ||
10. | ALA3426891 | (R)-9b | IC50 | = | 160 | nM | ALA3429146 | 6.80 | nM | Homo sapiens | ||
11. | ALA3426891 | (R)-9b | IC50 | = | 5 | nM | ALA3429145 | 8.30 | nM | Homo sapiens | ||
12. | ALA3426891 | (R)-9b | IC50 | = | 6 | nM | ALA3429144 | 8.22 | nM | Homo sapiens | ||
13. | ALA3426891 | (R)-9b | IC50 | = | 2 | uM | ALA3429143 | 5.70 | nM | |||
14. | ALA3426891 | (R)-9b | INH | 0 | ALA3429142 | Active | % | Homo sapiens | ||||
15. | ALA3426891 | (R)-9b | IC50 | = | 1.8 | uM | ALA3429141 | 5.75 | nM | Homo sapiens | ||
16. | ALA3426891 | (R)-9b | INH | = | 93.5 | % | ALA3429140 | % | Homo sapiens | |||
17. | ALA3426891 | (R)-9b | INH | = | 12.4 | % | ALA3428995 | % | Homo sapiens | |||
18. | ALA3426891 | (R)-9b | INH | = | 98.9 | % | ALA3428994 | % | Homo sapiens | |||
19. | ALA3426891 | (R)-9b | INH | = | 63.2 | % | ALA3428993 | % | Homo sapiens | |||
20. | ALA3426891 | (R)-9b | INH | = | 32 | % | ALA3428992 | % | Homo sapiens |