# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3527359 | YM150 monomaleate | Km | = | 27.3 | uM | ALA3538270 | nM | ||||
2. | ALA3527359 | YM150 monomaleate | Vmax | = | 0.608 | nmol/min | ALA3534350 | nmol/min | Homo sapiens | |||
3. | ALA3527359 | YM150 monomaleate | Ratio | = | 4.3 | ALA3538265 | ||||||
4. | ALA3527359 | YM150 monomaleate | CL free | = | 316 | uL/min/g | ALA3538264 | mL.min-1.g-1 | Homo sapiens | |||
5. | ALA3527359 | YM150 monomaleate | CL free | = | 257 | uL/min/g | ALA3538263 | mL.min-1.g-1 | Homo sapiens | |||
6. | ALA3527359 | YM150 monomaleate | CL free | = | 250 | uL/min/g | ALA3538262 | mL.min-1.g-1 | Homo sapiens | |||
7. | ALA3527359 | YM150 monomaleate | CL free | = | 138 | uL/min/g | ALA3538261 | mL.min-1.g-1 | Homo sapiens | |||
8. | ALA3527359 | YM150 monomaleate | Vmax | = | 5.79 | nmol/min | ALA3538260 | nmol/min | Homo sapiens | |||
9. | ALA3527359 | YM150 monomaleate | Vmax | = | 5.83 | nmol/min | ALA3538259 | nmol/min | Homo sapiens | |||
10. | ALA3527359 | YM150 monomaleate | Vmax | = | 5.59 | nmol/min | ALA3538258 | nmol/min | Homo sapiens | |||
11. | ALA3527359 | YM150 monomaleate | Vmax | = | 4.9 | nmol/min | ALA3537950 | nmol/min | Homo sapiens | |||
12. | ALA3527359 | YM150 monomaleate | Km(unbound) | = | 18.3 | uM | ALA3537949 | uM | Homo sapiens | |||
13. | ALA3527359 | YM150 monomaleate | Km(unbound) | = | 22.7 | uM | ALA3537948 | uM | Homo sapiens | |||
14. | ALA3527359 | YM150 monomaleate | Km(unbound) | = | 22.4 | uM | ALA3537947 | uM | Homo sapiens | |||
15. | ALA3527359 | YM150 monomaleate | Km(unbound) | = | 35.5 | uM | ALA3537946 | uM | Homo sapiens | |||
16. | ALA3527359 | YM150 monomaleate | CL free | = | 178 | uL/min/g | ALA3537945 | mL.min-1.g-1 | Homo sapiens | |||
17. | ALA3527359 | YM150 monomaleate | CL free | = | 184 | uL/min/g | ALA3537944 | mL.min-1.g-1 | Homo sapiens | |||
18. | ALA3527359 | YM150 monomaleate | CL free | = | 184 | uL/min/g | ALA3537943 | mL.min-1.g-1 | Homo sapiens | |||
19. | ALA3527359 | YM150 monomaleate | CL free | = | 17.4 | uL/min/g | ALA3537942 | mL.min-1.g-1 | Homo sapiens | |||
20. | ALA3527359 | YM150 monomaleate | Vmax | = | 3.14 | nmol/min | ALA3537941 | nmol/min | Homo sapiens |