# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3527524 | N-methyl-quinidine | INH | = | -6.1 | % | ALA2169429 | % | Homo sapiens | |||
2. | ALA3527524 | N-methyl-quinidine | INH | = | 21 | % | ALA2169430 | % | Homo sapiens | |||
3. | ALA3527524 | N-methyl-quinidine | INH | = | -10.3 | % | ALA2169431 | % | Homo sapiens | |||
4. | ALA3527524 | N-methyl-quinidine | Fu | = | 0.23 | ALA3537288 | Rattus norvegicus | |||||
5. | ALA3527524 | N-methyl-quinidine | Vdu | = | 4.6 | ml/g | ALA3537289 | L.kg-1 | Rattus norvegicus | |||
6. | ALA3527524 | N-methyl-quinidine | Kp | = | 1.06 | ALA3537290 | Rattus norvegicus | |||||
7. | ALA3527524 | N-methyl-quinidine | Compound recovery | 0 | ALA3537292 | Active | Rattus norvegicus | |||||
8. | ALA3527524 | N-methyl-quinidine | Compound recovery | 0 | ALA3537293 | Not Active | Rattus norvegicus | |||||
9. | ALA3527524 | N-methyl-quinidine | Compound recovery | 0 | ALA3537294 | Active | Rattus norvegicus | |||||
10. | ALA3527524 | N-methyl-quinidine | Activity | 0 | ALA2076302 | is not a substrate [-] | Rattus norvegicus | |||||
11. | ALA3527524 | N-methyl-quinidine | Activity | 0 | ALA2077578 | is not a substrate [-] | Rattus norvegicus | |||||
12. | ALA3527524 | N-methyl-quinidine | Km | = | 7.4 | uM | ALA2076040 | substrate [Km7.4uM] | nM | Rattus norvegicus | ||
13. | ALA3527524 | N-methyl-quinidine | Km | = | 12 | uM | ALA2076051 | substrate [Km12uM] | nM | Homo sapiens | ||
14. | ALA3527524 | N-methyl-quinidine | Km | = | 7.4 | uM | ALA2076040 | substrate [Km=7.4uM] | nM | Rattus norvegicus | ||
15. | ALA3527524 | N-methyl-quinidine | Km | = | 25.6 | uM | ALA2077577 | substrate [Km=25.6uM] | nM | Homo sapiens | ||
16. | ALA3527524 | N-methyl-quinidine | Activity | 0 | ALA2077102 | inhibitor [+] | Homo sapiens | |||||
17. | ALA3527524 | N-methyl-quinidine | Activity | 0 | ALA2076898 | inhibitor [+] | Rattus norvegicus | |||||
18. | ALA3527524 | N-methyl-quinidine | Activity | 0 | ALA2076307 | inhibitor [+] | Homo sapiens | |||||
19. | ALA3527524 | N-methyl-quinidine | Km | = | 11.5 | uM | ALA2076051 | substrate [Km=11.5uM] | nM | Homo sapiens |