# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3542370 | S-6-G, M0-2, Isoscutellarin | Drug uptake | 0 | ALA3533744 | Not Active | Homo sapiens | |||||
2. | ALA3542370 | S-6-G, M0-2, Isoscutellarin | Ki | = | 25.9 | uM | ALA3531160 | 4.59 | nM | Homo sapiens | ||
3. | ALA3542370 | S-6-G, M0-2, Isoscutellarin | Vmax/Km | = | 2.6 | microL/min/mg | ALA3531161 | microL/min/mg | Homo sapiens | |||
4. | ALA3542370 | S-6-G, M0-2, Isoscutellarin | Vmax | = | 19.7 | pmol/min/mg | ALA3531157 | pmol/min/mg | Homo sapiens | |||
5. | ALA3542370 | S-6-G, M0-2, Isoscutellarin | Km | = | 1.77 | uM | ALA3531157 | nM | Homo sapiens | |||
6. | ALA3542370 | S-6-G, M0-2, Isoscutellarin | Drug uptake | 0 | ALA3531156 | Active | Homo sapiens | |||||
7. | ALA3542370 | S-6-G, M0-2, Isoscutellarin | Drug uptake | 0 | ALA3533753 | Not Active | Homo sapiens | |||||
8. | ALA3542370 | S-6-G, M0-2, Isoscutellarin | Drug uptake | 0 | ALA3533752 | Not Active | Homo sapiens | |||||
9. | ALA3542370 | S-6-G, M0-2, Isoscutellarin | Drug uptake | 0 | ALA3533751 | Not Active | Homo sapiens | |||||
10. | ALA3542370 | S-6-G, M0-2, Isoscutellarin | Ratio | = | 20.4 | ALA3533750 | Homo sapiens | |||||
11. | ALA3542370 | S-6-G, M0-2, Isoscutellarin | Drug uptake | 0 | ALA3533749 | Not Active | Homo sapiens | |||||
12. | ALA3542370 | S-6-G, M0-2, Isoscutellarin | Ratio | = | 1.61 | ALA3533748 | Homo sapiens | |||||
13. | ALA3542370 | S-6-G, M0-2, Isoscutellarin | Ratio | = | 3.07 | ALA3533747 | Homo sapiens | |||||
14. | ALA3542370 | S-6-G, M0-2, Isoscutellarin | Ratio | = | 57.5 | ALA3533746 | Homo sapiens | |||||
15. | ALA3542370 | S-6-G, M0-2, Isoscutellarin | INH | 0 | ALA3533745 | Active | % | Homo sapiens | ||||
16. | ALA3542370 | S-6-G, M0-2, Isoscutellarin | INH | 0 | ALA3536906 | Active | % | Homo sapiens | ||||
17. | ALA3542370 | S-6-G, M0-2, Isoscutellarin | INH | 0 | ALA3536905 | Active | % | Homo sapiens | ||||
18. | ALA3542370 | S-6-G, M0-2, Isoscutellarin | IC50 | = | 20 | uM | ALA3536904 | 4.70 | nM | Homo sapiens | ||
19. | ALA3542370 | S-6-G, M0-2, Isoscutellarin | IC50 | = | 50 | uM | ALA3536903 | 4.30 | nM | Homo sapiens | ||
20. | ALA3542370 | S-6-G, M0-2, Isoscutellarin | Vmax/Km | = | 2.84 | microL/min/mg | ALA3536902 | microL/min/mg | Homo sapiens |