| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3582472 | 26 | INH | 0 | ALA3583963 | Not Active | % | Rattus norvegicus | ||||
| 2. | ALA3582472 | 26 | INH | 0 | ALA3583962 | Active | % | |||||
| 3. | ALA3582472 | 26 | t1/2 | = | 7.4 | hr | ALA3583961 | hr | Macaca mulatta | |||
| 4. | ALA3582472 | 26 | CL | = | 10 | ml/min.kg | ALA3583960 | mL.min-1.kg-1 | Macaca mulatta | |||
| 5. | ALA3582472 | 26 | AUC/dose | = | 3.07 | uM.hr.kg/mg | ALA3583959 | uM.hr.kg/mg | Macaca mulatta | |||
| 6. | ALA3582472 | 26 | F | = | 53 | % | ALA3583958 | % | Macaca mulatta | |||
| 7. | ALA3582472 | 26 | CLH | < | 20 | ml/min.kg | ALA3583957 | mL.min-1.kg-1 | ||||
| 8. | ALA3582472 | 26 | Fu | = | 23 | % | ALA3583956 | Macaca mulatta | ||||
| 9. | ALA3582472 | 26 | IC50 | > | 30 | uM | ALA3583955 | nM | Homo sapiens | |||
| 10. | ALA3582472 | 26 | IC50 | > | 30 | uM | ALA3583954 | nM | Homo sapiens | |||
| 11. | ALA3582472 | 26 | IC50 | = | 2.49 | uM | ALA3583953 | 5.60 | nM | Homo sapiens | ||
| 12. | ALA3582472 | 26 | Ratio IC50 | = | 500 | ALA3583949 | ||||||
| 13. | ALA3582472 | 26 | INH | 0 | ALA3583948 | Not Active | % | Homo sapiens | ||||
| 14. | ALA3582472 | 26 | INH | 0 | ALA3583947 | Not Active | % | Homo sapiens | ||||
| 15. | ALA3582472 | 26 | IC50 | > | 50000 | nM | ALA3583946 | nM | Homo sapiens | |||
| 16. | ALA3582472 | 26 | IC50 | > | 10000 | nM | ALA3583945 | nM | Homo sapiens | |||
| 17. | ALA3582472 | 26 | IC50 | = | 4513 | nM | ALA3583830 | 5.35 | nM | Homo sapiens | ||
| 18. | ALA3582472 | 26 | IC50 | > | 10000 | nM | ALA3583829 | nM | Homo sapiens | |||
| 19. | ALA3582472 | 26 | CL | = | 37 | ml/min.kg | ALA3583944 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 20. | ALA3582472 | 26 | AUC/dose | = | 2.1 | uM.hr.kg/mg | ALA3583943 | uM.hr.kg/mg | Rattus norvegicus |
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