# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3586432 | 30 | Ki | = | 12 | nM | ALA3587482 | 7.92 | nM | Homo sapiens | ||
2. | ALA3586432 | 30 | Kb | = | 3.5 | nM | ALA3587482 | nM | Homo sapiens | |||
3. | ALA3586432 | 30 | Cmax | = | 148 | ng/ml | ALA3587722 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
4. | ALA3586432 | 30 | F | = | 8 | % | ALA3587710 | % | Rattus norvegicus | |||
5. | ALA3586432 | 30 | t1/2 | = | 0.27 | hr | ALA3587709 | hr | Rattus norvegicus | |||
6. | ALA3586432 | 30 | Vdss | = | 0.7 | L/Kg | ALA3587708 | L.kg-1 | Rattus norvegicus | |||
7. | ALA3586432 | 30 | CL | = | 52.1 | ml/min.kg | ALA3587707 | mL.min-1.kg-1 | Rattus norvegicus | |||
8. | ALA3586432 | 30 | Occ | = | 67 | % | ALA3587705 | % | Rattus norvegicus | |||
9. | ALA3586432 | 30 | Ki | = | 2 | nM | ALA3587703 | 8.70 | nM | Rattus norvegicus | ||
10. | ALA3586432 | 30 | IC50 | > | 10 | uM | ALA3587702 | nM | Homo sapiens | |||
11. | ALA3586432 | 30 | ERH | = | 0.87 | ALA3587701 | Homo sapiens | |||||
12. | ALA3586432 | 30 | ERH | = | 0.79 | ALA3587700 | Rattus norvegicus | |||||
13. | ALA3586432 | 30 | Ki | = | 1640 | nM | ALA3587483 | 5.79 | nM | Homo sapiens |