# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3586433 | 31 | Ki | = | 14 | nM | ALA3587482 | 7.85 | nM | Homo sapiens | ||
2. | ALA3586433 | 31 | Kb | = | 2.9 | nM | ALA3587482 | nM | Homo sapiens | |||
3. | ALA3586433 | 31 | IC50 | = | 3.1 | uM | ALA3587716 | 5.51 | nM | Homo sapiens | ||
4. | ALA3586433 | 31 | PB | = | 84.4 | % | ALA3587715 | % | Rattus norvegicus | |||
5. | ALA3586433 | 31 | PPB | = | 72.7 | % | ALA3587714 | % | Rattus norvegicus | |||
6. | ALA3586433 | 31 | PPB | = | 90.5 | % | ALA3587713 | % | Homo sapiens | |||
7. | ALA3586433 | 31 | Papp | = | 49.7 | ucm/s | ALA3587711 | ucm/s | Homo sapiens | |||
8. | ALA3586433 | 31 | Papp | = | 62.3 | ucm/s | ALA3587712 | ucm/s | Homo sapiens | |||
9. | ALA3586433 | 31 | F | = | 21 | % | ALA3587710 | % | Rattus norvegicus | |||
10. | ALA3586433 | 31 | t1/2 | = | 0.2 | hr | ALA3587709 | hr | Rattus norvegicus | |||
11. | ALA3586433 | 31 | Vdss | = | 0.7 | L/Kg | ALA3587708 | L.kg-1 | Rattus norvegicus | |||
12. | ALA3586433 | 31 | CL | = | 57 | ml/min.kg | ALA3587707 | mL.min-1.kg-1 | Rattus norvegicus | |||
13. | ALA3586433 | 31 | Occ | = | 49 | % | ALA3587706 | % | Rattus norvegicus | |||
14. | ALA3586433 | 31 | Ki | = | 10 | nM | ALA3587703 | 8.00 | nM | Rattus norvegicus | ||
15. | ALA3586433 | 31 | IC50 | = | 6 | uM | ALA3587702 | 5.22 | nM | Homo sapiens | ||
16. | ALA3586433 | 31 | ERH | = | 0.83 | ALA3587701 | Homo sapiens | |||||
17. | ALA3586433 | 31 | ERH | = | 0.71 | ALA3587700 | Rattus norvegicus | |||||
18. | ALA3586433 | 31 | Ki | = | 2280 | nM | ALA3587483 | 5.64 | nM | Homo sapiens |