# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3586434 | 32 | Ki | = | 10 | nM | ALA3587482 | 8.00 | nM | Homo sapiens | ||
2. | ALA3586434 | 32 | Kb | = | 5.3 | nM | ALA3587482 | nM | Homo sapiens | |||
3. | ALA3586434 | 32 | IC50 | = | 9.3 | uM | ALA3587716 | 5.03 | nM | Homo sapiens | ||
4. | ALA3586434 | 32 | PB | 0 | ALA3587715 | Not Determined | % | Rattus norvegicus | ||||
5. | ALA3586434 | 32 | PPB | = | 88.4 | % | ALA3587714 | % | Rattus norvegicus | |||
6. | ALA3586434 | 32 | PPB | = | 92.5 | % | ALA3587713 | % | Homo sapiens | |||
7. | ALA3586434 | 32 | Papp | = | 26.8 | ucm/s | ALA3587711 | ucm/s | Homo sapiens | |||
8. | ALA3586434 | 32 | Papp | = | 58.1 | ucm/s | ALA3587712 | ucm/s | Homo sapiens | |||
9. | ALA3586434 | 32 | F | = | 18 | % | ALA3587710 | % | Rattus norvegicus | |||
10. | ALA3586434 | 32 | t1/2 | = | 0.37 | hr | ALA3587709 | hr | Rattus norvegicus | |||
11. | ALA3586434 | 32 | Vdss | = | 1.5 | L/Kg | ALA3587708 | L.kg-1 | Rattus norvegicus | |||
12. | ALA3586434 | 32 | CL | = | 65.5 | ml/min.kg | ALA3587707 | mL.min-1.kg-1 | Rattus norvegicus | |||
13. | ALA3586434 | 32 | Occ | = | 72 | % | ALA3587705 | % | Rattus norvegicus | |||
14. | ALA3586434 | 32 | Ki | = | 14 | nM | ALA3587703 | 7.85 | nM | Rattus norvegicus | ||
15. | ALA3586434 | 32 | IC50 | > | 10 | uM | ALA3587702 | nM | Homo sapiens | |||
16. | ALA3586434 | 32 | ERH | = | 0.88 | ALA3587701 | Homo sapiens | |||||
17. | ALA3586434 | 32 | ERH | = | 0.82 | ALA3587700 | Rattus norvegicus | |||||
18. | ALA3586434 | 32 | Ki | = | 1960 | nM | ALA3587483 | 5.71 | nM | Homo sapiens |