# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3586443 | 7 | INH | = | 86 | % | ALA5252738 | % | Homo sapiens | |||
2. | ALA3586443 | 7 | INH | = | 94.4 | % | ALA5252737 | % | Homo sapiens | |||
3. | ALA3586443 | 7 | INH | = | 12 | % | ALA5252736 | % | Homo sapiens | |||
4. | ALA3586443 | 7 | INH | = | 15 | % | ALA5252735 | % | Homo sapiens | |||
5. | ALA3586443 | 7 | INH | = | 1 | % | ALA5252734 | % | Homo sapiens | |||
6. | ALA3586443 | 7 | INH | = | 48 | % | ALA5252705 | % | Homo sapiens | |||
7. | ALA3586443 | 7 | EC50 | > | 50 | uM | ALA3588237 | nM | Homo sapiens | |||
8. | ALA3586443 | 7 | IC50 | = | 13 | uM | ALA3588238 | 4.89 | nM | Homo sapiens | ||
9. | ALA3586443 | 7 | ERH | = | 0.77 | ALA3588239 | Homo sapiens | |||||
10. | ALA3586443 | 7 | ERH | = | 0.5 | ALA3588240 | Rattus norvegicus | |||||
11. | ALA3586443 | 7 | Papp | = | 288 | nm/s | ALA3588241 | nm/s | Sus scrofa | |||
12. | ALA3586443 | 7 | Ratio | = | 0.7 | ALA3588242 | Sus scrofa | |||||
13. | ALA3586443 | 7 | CL | = | 22 | ml/min.kg | ALA3588243 | mL.min-1.kg-1 | Rattus norvegicus | |||
14. | ALA3586443 | 7 | ERH | = | 0.3 | ALA3588244 | Rattus norvegicus | |||||
15. | ALA3586443 | 7 | Vdss | = | 0.7 | L/Kg | ALA3588245 | L.kg-1 | Rattus norvegicus | |||
16. | ALA3586443 | 7 | t1/2 | = | 1.3 | hr | ALA3588246 | hr | Rattus norvegicus | |||
17. | ALA3586443 | 7 | F | = | 35 | % | ALA3588247 | % | Rattus norvegicus | |||
18. | ALA3586443 | 7 | IC50 | = | 240 | uM | ALA3588253 | 3.62 | nM | Homo sapiens |