# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3589001 | 4 | Stability | 0 | ALA3592361 | Stable | % | Rattus norvegicus | ||||
2. | ALA3589001 | 4 | Stability | 0 | ALA3592360 | Unstable | % | Rattus norvegicus | ||||
3. | ALA3589001 | 4 | Stability | 0 | ALA3592357 | Unstable | % | Mus musculus | ||||
4. | ALA3589001 | 4 | Retention_time | = | 23.6 | min | ALA3592352 | min | Mus musculus | |||
5. | ALA3589001 | 4 | Activity | 0 | ALA3592351 | Non-toxic | Homo sapiens | |||||
6. | ALA3589001 | 4 | Activity | > | 80 | % | ALA3592350 | % | Homo sapiens | |||
7. | ALA3589001 | 4 | t1/2 | = | 3.43 | hr | ALA3592349 | hr | Mus musculus | |||
8. | ALA3589001 | 4 | t1/2 | = | 6 | hr | ALA3592348 | hr | Homo sapiens | |||
9. | ALA3589001 | 4 | Ratio | = | 9.2 | ALA3592347 | ||||||
10. | ALA3589001 | 4 | Ki(app) | = | 18.3 | nM | ALA3592346 | 7.74 | nM | Homo sapiens | ||
11. | ALA3589001 | 4 | Ki | = | 2 | nM | ALA3592345 | 8.70 | nM | Homo sapiens |