| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3588871 | (S)-9a | Stability | = | 4 | % | ALA4135892 | % | ||||
| 2. | ALA3588871 | (S)-9a | EC50 | = | 0.086 | uM | ALA4135891 | 7.07 | nM | Homo sapiens | ||
| 3. | ALA3588871 | (S)-9a | EC50 | = | 0.26 | uM | ALA4135888 | 6.58 | nM | Homo sapiens | ||
| 4. | ALA3588871 | (S)-9a | EC50 | = | 0.19 | uM | ALA4135886 | 6.72 | nM | Homo sapiens | ||
| 5. | ALA3588871 | (S)-9a | CLH | = | 1162.4 | microL/min/mg | ALA3592690 | mL.min-1.g-1 | Rattus norvegicus | |||
| 6. | ALA3588871 | (S)-9a | t1/2 | = | 1.1 | min | ALA3592689 | hr | Rattus norvegicus | |||
| 7. | ALA3588871 | (S)-9a | Efficacy | = | 110 | % | ALA3592688 | % | Mus musculus | |||
| 8. | ALA3588871 | (S)-9a | EC50 | = | 0.24 | uM | ALA3592687 | 6.62 | nM | Mus musculus | ||
| 9. | ALA3588871 | (S)-9a | Efficacy | = | 105 | % | ALA3592686 | % | Homo sapiens | |||
| 10. | ALA3588871 | (S)-9a | Efficacy | = | 100 | % | ALA3592685 | % | Homo sapiens | |||
| 11. | ALA3588871 | (S)-9a | EC50 | = | 0.06 | uM | ALA3592684 | 7.22 | nM | Homo sapiens | ||
| 12. | ALA3588871 | (S)-9a | Efficacy | = | 120 | % | ALA3592682 | % | Homo sapiens | |||
| 13. | ALA3588871 | (S)-9a | Efficacy | = | 130 | % | ALA3592681 | % | Homo sapiens | |||
| 14. | ALA3588871 | (S)-9a | EC50 | = | 0.096 | uM | ALA3592680 | 7.02 | nM | Homo sapiens | ||
| 15. | ALA3588871 | (S)-9a | EC50 | = | 0.43 | uM | ALA3592565 | 6.37 | nM | Homo sapiens | ||
| 16. | ALA3588871 | (S)-9a | EC50 | = | 0.064 | uM | ALA3592683 | 7.19 | nM | Homo sapiens |
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