# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3589946 | (R)-9a | CLH | = | 1290.6 | microL/min/mg | ALA3592690 | mL.min-1.g-1 | Rattus norvegicus | |||
2. | ALA3589946 | (R)-9a | t1/2 | = | 1.2 | min | ALA3592689 | hr | Rattus norvegicus | |||
3. | ALA3589946 | (R)-9a | Efficacy | = | 30 | % | ALA3592688 | % | Mus musculus | |||
4. | ALA3589946 | (R)-9a | EC50 | = | 4.9 | uM | ALA3592687 | 5.31 | nM | Mus musculus | ||
5. | ALA3589946 | (R)-9a | Efficacy | = | 95 | % | ALA3592686 | % | Homo sapiens | |||
6. | ALA3589946 | (R)-9a | Efficacy | = | 40 | % | ALA3592685 | % | Homo sapiens | |||
7. | ALA3589946 | (R)-9a | EC50 | = | 0.88 | uM | ALA3592684 | 6.06 | nM | Homo sapiens | ||
8. | ALA3589946 | (R)-9a | Efficacy | = | 100 | % | ALA3592682 | % | Homo sapiens | |||
9. | ALA3589946 | (R)-9a | EC50 | = | 0.23 | uM | ALA3592680 | 6.64 | nM | Homo sapiens | ||
10. | ALA3589946 | (R)-9a | EC50 | 0 | ALA3592565 | Not Active | Homo sapiens | |||||
11. | ALA3589946 | (R)-9a | EC50 | = | 0.92 | uM | ALA3592683 | 6.04 | nM | Homo sapiens |