# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3590120 | 12 | t1/2 | = | 120 | hr | ALA3591271 | hr | Mus musculus | |||
2. | ALA3590120 | 12 | t1/2 | = | 54 | hr | ALA3591270 | hr | Mus musculus | |||
3. | ALA3590120 | 12 | Stability | 0 | ALA3591268 | Stable | % | |||||
4. | ALA3590120 | 12 | t1/2 | = | 42 | min | ALA3591267 | hr | ||||
5. | ALA3590120 | 12 | INH | 0 | ALA3591264 | Active | % | Homo sapiens | ||||
6. | ALA3590120 | 12 | INH | 0 | ALA3591263 | Active | % | Homo sapiens | ||||
7. | ALA3590120 | 12 | CLH | > | 250 | microL/min/mg | ALA3591261 | mL.min-1.g-1 | ||||
8. | ALA3590120 | 12 | CLH | = | 13 | microL/min/mg | ALA3591260 | mL.min-1.g-1 | Homo sapiens | |||
9. | ALA3590120 | 12 | Selectivity ratio | = | 2 | ALA3593143 | ||||||
10. | ALA3590120 | 12 | Selectivity ratio | = | 2 | ALA3593142 | ||||||
11. | ALA3590120 | 12 | solubility | = | 150 | uM | ALA3593141 | nM | ||||
12. | ALA3590120 | 12 | logD | = | 2.3 | ALA3593140 | ||||||
13. | ALA3590120 | 12 | IC50 | > | 10 | uM | ALA3593139 | nM | Homo sapiens | |||
14. | ALA3590120 | 12 | IC50 | = | 0.041 | uM | ALA3593138 | 7.39 | nM | Homo sapiens | ||
15. | ALA3590120 | 12 | IC50 | = | 0.028 | uM | ALA3593137 | 7.55 | nM | Homo sapiens | ||
16. | ALA3590120 | 12 | IC50 | = | 0.003 | uM | ALA3593134 | 8.51 | nM | Homo sapiens | ||
17. | ALA3590120 | 12 | IC50 | = | 0.003 | uM | ALA3593135 | 8.52 | nM | Homo sapiens | ||
18. | ALA3590120 | 12 | IC50 | = | 0.007 | uM | ALA3593136 | 8.17 | nM | Homo sapiens |