# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3597624 | 25 | Stability | 0 | ALA3599410 | Stable | % | |||||
2. | ALA3597624 | 25 | Stability | 0 | ALA3599409 | Stable | % | |||||
3. | ALA3597624 | 25 | Stability | 0 | ALA3599408 | Stable | % | |||||
4. | ALA3597624 | 25 | INH | = | 25 | % | ALA3599290 | % | Cavia porcellus | |||
5. | ALA3597624 | 25 | INH | = | 57 | % | ALA3599289 | % | Cavia porcellus | |||
6. | ALA3597624 | 25 | IC50 | = | 24 | nM | ALA3599288 | 7.62 | nM | Cavia porcellus | ||
7. | ALA3597624 | 25 | IC50 | = | 2.2 | nM | ALA3599287 | 8.66 | nM | Cavia porcellus | ||
8. | ALA3597624 | 25 | F | = | 66 | % | ALA3599286 | % | Cavia porcellus | |||
9. | ALA3597624 | 25 | AUC | = | 10.5 | microg.hr/mL | ALA3599285 | ng.hr.mL-1 | Cavia porcellus | |||
10. | ALA3597624 | 25 | INH | = | 97 | % | ALA3599284 | % | Cavia porcellus | |||
11. | ALA3597624 | 25 | INH | = | 96 | % | ALA3599268 | % | Cavia porcellus | |||
12. | ALA3597624 | 25 | Papp | = | 7.9 | ucm/s | ALA3599264 | ucm/s | ||||
13. | ALA3597624 | 25 | IC50 | = | 5.5 | nM | ALA3599261 | 8.26 | nM | Homo sapiens | ||
14. | ALA3597624 | 25 | IC50 | = | 1.5 | nM | ALA3599260 | 8.82 | nM | Homo sapiens |