| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3600453 | 8c, 2-Pyz-L-His(2,5-dibromo)-L-ProNH2 | Time | = | 96 | s | ALA3602713 | hr | Rattus norvegicus | |||
| 2. | ALA3600453 | 8c, 2-Pyz-L-His(2,5-dibromo)-L-ProNH2 | Time | = | 167 | s | ALA3602712 | hr | Rattus norvegicus | |||
| 3. | ALA3600453 | 8c, 2-Pyz-L-His(2,5-dibromo)-L-ProNH2 | Activity | 0 | ALA3602711 | Active | Rattus norvegicus | |||||
| 4. | ALA3600453 | 8c, 2-Pyz-L-His(2,5-dibromo)-L-ProNH2 | Activity | 0 | ALA3602710 | Active | Rattus norvegicus | |||||
| 5. | ALA3600453 | 8c, 2-Pyz-L-His(2,5-dibromo)-L-ProNH2 | Time | = | 36.31 | s | ALA3602709 | hr | Rattus norvegicus | |||
| 6. | ALA3600453 | 8c, 2-Pyz-L-His(2,5-dibromo)-L-ProNH2 | Activity | = | 2.25 | ALA3602708 | Rattus norvegicus | |||||
| 7. | ALA3600453 | 8c, 2-Pyz-L-His(2,5-dibromo)-L-ProNH2 | Activity | 0 | ALA3602707 | Active | Rattus norvegicus | |||||
| 8. | ALA3600453 | 8c, 2-Pyz-L-His(2,5-dibromo)-L-ProNH2 | Activity | 0 | ALA3602706 | Non-toxic | Rattus norvegicus | |||||
| 9. | ALA3600453 | 8c, 2-Pyz-L-His(2,5-dibromo)-L-ProNH2 | Activity | 0 | ALA3602677 | Active | Rattus norvegicus | |||||
| 10. | ALA3600453 | 8c, 2-Pyz-L-His(2,5-dibromo)-L-ProNH2 | Activity | = | 196.08 | mm3 | ALA3602676 | mm3 | Rattus norvegicus | |||
| 11. | ALA3600453 | 8c, 2-Pyz-L-His(2,5-dibromo)-L-ProNH2 | Stability | 0 | ALA3602675 | Stable | % | Mus musculus | ||||
| 12. | ALA3600453 | 8c, 2-Pyz-L-His(2,5-dibromo)-L-ProNH2 | Cp | = | 5.31 | ng/ml | ALA3602670 | ng/ml | Rattus norvegicus | |||
| 13. | ALA3600453 | 8c, 2-Pyz-L-His(2,5-dibromo)-L-ProNH2 | Cp | = | 5.15 | ng/ml | ALA3602669 | ng/ml | Rattus norvegicus | |||
| 14. | ALA3600453 | 8c, 2-Pyz-L-His(2,5-dibromo)-L-ProNH2 | Cp | = | 4.85 | ng/ml | ALA3602668 | ng/ml | Rattus norvegicus | |||
| 15. | ALA3600453 | 8c, 2-Pyz-L-His(2,5-dibromo)-L-ProNH2 | INH | = | 74.8 | % | ALA3602667 | % | Mus musculus | |||
| 16. | ALA3600453 | 8c, 2-Pyz-L-His(2,5-dibromo)-L-ProNH2 | Ratio EC50 | = | 50.8 | ALA3602666 | ||||||
| 17. | ALA3600453 | 8c, 2-Pyz-L-His(2,5-dibromo)-L-ProNH2 | EC50 | = | 0.05 | uM | ALA3602665 | 7.30 | nM | Mus musculus | ||
| 18. | ALA3600453 | 8c, 2-Pyz-L-His(2,5-dibromo)-L-ProNH2 | IC50 | > | 50 | uM | ALA3602662 | nM | Mus musculus | |||
| 19. | ALA3600453 | 8c, 2-Pyz-L-His(2,5-dibromo)-L-ProNH2 | IC50 | > | 50 | uM | ALA3602663 | nM | Mus musculus | |||
| 20. | ALA3600453 | 8c, 2-Pyz-L-His(2,5-dibromo)-L-ProNH2 | EC50 | = | 2.54 | uM | ALA3602664 | 5.59 | nM | Mus musculus |
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