# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3604734 | 1ah | Activity | = | 198 | % | ALA3607764 | % | Mus musculus | |||
2. | ALA3604734 | 1ah | Activity | = | 283 | % | ALA3607763 | % | Mus musculus | |||
3. | ALA3604734 | 1ah | Activity | = | 595 | % | ALA3607762 | % | Mus musculus | |||
4. | ALA3604734 | 1ah | IC50 | = | 510 | nM | ALA3607749 | 6.29 | nM | Homo sapiens | ||
5. | ALA3604734 | 1ah | IC50 | = | 115 | nM | ALA3607750 | 6.94 | nM | Mus musculus | ||
6. | ALA3604734 | 1ah | permeability | = | 420 | nm/s | ALA3607751 | nm/s | ||||
7. | ALA3604734 | 1ah | solubility | = | 0.095 | mg/ml | ALA3607752 | ug.mL-1 | ||||
8. | ALA3604734 | 1ah | pIC50 | = | 4.9 | ALA3607753 | 4.90 | nM | Homo sapiens | |||
9. | ALA3604734 | 1ah | t1/2 | > | 90 | min | ALA3607754 | hr | Mus musculus | |||
10. | ALA3604734 | 1ah | pIC50 | = | 6.4 | ALA3607755 | 6.40 | nM | Homo sapiens | |||
11. | ALA3604734 | 1ah | beta t1/2 | = | 4.1 | hr | ALA3607756 | hr | Mus musculus | |||
12. | ALA3604734 | 1ah | CL | = | 24 | ml/min.kg | ALA3607757 | mL.min-1.kg-1 | Mus musculus | |||
13. | ALA3604734 | 1ah | Vdss | = | 6.4 | L/Kg | ALA3607758 | L.kg-1 | Mus musculus | |||
14. | ALA3604734 | 1ah | F | = | 35 | % | ALA3607759 | % | Mus musculus | |||
15. | ALA3604734 | 1ah | AUC/dose | = | 260 | ng/hr/ml | ALA3607760 | ng/hr/ml | Mus musculus | |||
16. | ALA3604734 | 1ah | Activity | = | 1483 | % | ALA3607761 | % | Mus musculus | |||
17. | ALA3604734 | 1ah | logD | = | 5.1 | ALA4222838 | ||||||
18. | ALA3604734 | 1ah | pIC50 | = | 4.9 | ALA4222830 | 4.90 | nM | Homo sapiens | |||
19. | ALA3604734 | 1ah | pIC50 | = | 6.4 | ALA4222828 | 6.40 | nM | Homo sapiens | |||
20. | ALA3604734 | 1ah | IC50 | = | 510 | nM | ALA4222829 | 6.29 | nM | Homo sapiens |