| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3608740 | 17 | IC50 | = | 50000 | nM | ALA3888930 | 4.30 | 423448 | nM | Homo sapiens | |
| 2. | ALA3608740 | 17 | Ki | > | 30000 | nM | ALA3888929 | 423406 | nM | Homo sapiens | ||
| 3. | ALA3608740 | 17 | Ki | > | 30000 | nM | ALA3888928 | 423362 | nM | Homo sapiens | ||
| 4. | ALA3608740 | 17 | Ki | = | 60 | nM | ALA3888927 | 7.22 | 423316 | nM | Homo sapiens | |
| 5. | ALA3608740 | 17 | IC50 | = | 93 | nM | ALA3888926 | 7.03 | 423269 | nM | Homo sapiens | |
| 6. | ALA3608740 | 17 | Ratio | = | 0.26 | ALA3610294 | ||||||
| 7. | ALA3608740 | 17 | Ratio | = | 1.58 | ALA3610292 | ||||||
| 8. | ALA3608740 | 17 | Ratio | = | 7.71 | ALA3610115 | ||||||
| 9. | ALA3608740 | 17 | Ratio | = | 47.3 | ALA3610113 | ||||||
| 10. | ALA3608740 | 17 | Tmax | = | 45 | min | ALA3610111 | hr | Rattus norvegicus | |||
| 11. | ALA3608740 | 17 | MED | = | 30 | mg kg-1 | ALA3610109 | mg kg-1 | Rattus norvegicus | |||
| 12. | ALA3608740 | 17 | Ki | = | 573 | nM | ALA3610107 | 6.24 | nM | Rattus norvegicus | ||
| 13. | ALA3608740 | 17 | F | = | 55 | % | ALA3610105 | % | Rattus norvegicus | |||
| 14. | ALA3608740 | 17 | t1/2 | = | 35 | min | ALA3610103 | hr | Rattus norvegicus | |||
| 15. | ALA3608740 | 17 | Vdss | = | 0.68 | L/Kg | ALA3610101 | L.kg-1 | Rattus norvegicus | |||
| 16. | ALA3608740 | 17 | CL | = | 13.7 | min/ml/kg | ALA3610099 | min/ml/kg | Rattus norvegicus | |||
| 17. | ALA3608740 | 17 | BPR | = | 0.17 | ALA3610098 | ||||||
| 18. | ALA3608740 | 17 | Drug uptake(free) | = | 68.6 | nM | ALA3610097 | nM | Rattus norvegicus | |||
| 19. | ALA3608740 | 17 | Cp(f) | = | 406.7 | nM | ALA3610095 | nM | Rattus norvegicus | |||
| 20. | ALA3608740 | 17 | Fu | = | 0.604 | ALA3610094 | Rattus norvegicus |
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