# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3629181 | 2a,b, diastereomeric mixture | INH | > | 40 | % | ALA3632405 | % | Trypanosoma brucei rhodesiense | |||
2. | ALA3629181 | 2a,b, diastereomeric mixture | INH | 0 | ALA3632406 | Not Active | % | Homo sapiens | ||||
3. | ALA3629181 | 2a,b, diastereomeric mixture | INH | 0 | ALA3632407 | Not Active | % | Homo sapiens | ||||
4. | ALA3629181 | 2a,b, diastereomeric mixture | IC50 | = | 16.45 | uM | ALA3632408 | 4.78 | nM | Trypanosoma brucei brucei | ||
5. | ALA3629181 | 2a,b, diastereomeric mixture | IC50 | = | 18.2 | uM | ALA3632409 | 4.74 | nM | Trypanosoma brucei brucei | ||
6. | ALA3629181 | 2a,b, diastereomeric mixture | IC50 | > | 100 | uM | ALA3632410 | nM | ||||
7. | ALA3629181 | 2a,b, diastereomeric mixture | Ki | = | 8.41 | uM | ALA3632411 | 5.08 | nM | Trypanosoma brucei rhodesiense |