| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3633248 | 5 | pKinact | = | 2.41 | ALA3636509 | Homo sapiens | |||||
| 2. | ALA3633248 | 5 | F | = | 31 | % | ALA3636545 | % | Canis lupus familiaris | |||
| 3. | ALA3633248 | 5 | F | = | 76 | % | ALA3636544 | % | Rattus norvegicus | |||
| 4. | ALA3633248 | 5 | Tmax | = | 1.5 | hr | ALA3636541 | hr | Canis lupus familiaris | |||
| 5. | ALA3633248 | 5 | Tmax | = | 0.5 | hr | ALA3636540 | hr | Rattus norvegicus | |||
| 6. | ALA3633248 | 5 | beta t1/2 | = | 3.4 | hr | ALA3636537 | hr | Canis lupus familiaris | |||
| 7. | ALA3633248 | 5 | beta t1/2 | = | 0.76 | hr | ALA3636536 | hr | Rattus norvegicus | |||
| 8. | ALA3633248 | 5 | Vdss | = | 0.3 | L/Kg | ALA3636533 | L.kg-1 | Canis lupus familiaris | |||
| 9. | ALA3633248 | 5 | Vdss | = | 1.23 | L/Kg | ALA3636532 | L.kg-1 | Rattus norvegicus | |||
| 10. | ALA3633248 | 5 | CL | = | 1.31 | ml/min.kg | ALA3636529 | mL.min-1.kg-1 | Canis lupus familiaris | |||
| 11. | ALA3633248 | 5 | CL | = | 35.1 | ml/min.kg | ALA3636528 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 12. | ALA3633248 | 5 | CLH(app) | < | 6 | uL/min | ALA3636527 | uL/min | Homo sapiens | |||
| 13. | ALA3633248 | 5 | CLH(app) | < | 8 | uL/min/ug | ALA3636526 | mL.min-1.g-1 | Homo sapiens | |||
| 14. | ALA3633248 | 5 | Fu | = | 0.5 | ALA3636525 | Homo sapiens | |||||
| 15. | ALA3633248 | 5 | Papp | = | 0.8 | ucm/s | ALA3636521 | ucm/s | ||||
| 16. | ALA3633248 | 5 | IC50 | = | 2.6 | uM | ALA3636511 | 5.58 | nM | Homo sapiens | ||
| 17. | ALA3633248 | 5 | log(ratio) | = | 4.03 | ALA3636510 | Homo sapiens | |||||
| 18. | ALA3633248 | 5 | pKi | = | 6.43 | ALA3636509 | 6.43 | nM | Homo sapiens | |||
| 19. | ALA3633248 | 5 | logD | = | 0.59 | ALA3636508 | ||||||
| 20. | ALA3633248 | 5 | Ratio | = | 15 | ALA3636507 | Homo sapiens |
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