| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA3633250 | 4 | pKinact | = | 2.61 | ALA3636509 | Homo sapiens | |||||
| 2. | ALA3633250 | 4 | F | = | 84 | % | ALA3636545 | % | Canis lupus familiaris | |||
| 3. | ALA3633250 | 4 | F | = | 91 | % | ALA3636544 | % | Rattus norvegicus | |||
| 4. | ALA3633250 | 4 | Tmax | = | 1.3 | hr | ALA3636541 | hr | Canis lupus familiaris | |||
| 5. | ALA3633250 | 4 | Tmax | = | 0.38 | hr | ALA3636540 | hr | Rattus norvegicus | |||
| 6. | ALA3633250 | 4 | beta t1/2 | = | 5.7 | hr | ALA3636537 | hr | Canis lupus familiaris | |||
| 7. | ALA3633250 | 4 | beta t1/2 | = | 1.1 | hr | ALA3636536 | hr | Rattus norvegicus | |||
| 8. | ALA3633250 | 4 | Vdss | = | 3.66 | L/Kg | ALA3636533 | L.kg-1 | Canis lupus familiaris | |||
| 9. | ALA3633250 | 4 | Vdss | = | 3.71 | L/Kg | ALA3636532 | L.kg-1 | Rattus norvegicus | |||
| 10. | ALA3633250 | 4 | CL | = | 13.4 | ml/min.kg | ALA3636529 | mL.min-1.kg-1 | Canis lupus familiaris | |||
| 11. | ALA3633250 | 4 | CL | = | 70.3 | ml/min.kg | ALA3636528 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 12. | ALA3633250 | 4 | CLH(app) | = | 2.9 | uL/min | ALA3636527 | uL/min | Homo sapiens | |||
| 13. | ALA3633250 | 4 | CLH(app) | = | 8.8 | uL/min/ug | ALA3636526 | mL.min-1.g-1 | Homo sapiens | |||
| 14. | ALA3633250 | 4 | Fu | = | 0.7 | ALA3636525 | Homo sapiens | |||||
| 15. | ALA3633250 | 4 | Papp | = | 3.5 | ucm/s | ALA3636521 | ucm/s | ||||
| 16. | ALA3633250 | 4 | Drug metabolism | 0 | ALA3636524 | metabolite_notdetected | ||||||
| 17. | ALA3633250 | 4 | IC50 | = | 0.5 | uM | ALA3636511 | 6.30 | nM | Homo sapiens | ||
| 18. | ALA3633250 | 4 | log(ratio) | = | 4.13 | ALA3636510 | Homo sapiens | |||||
| 19. | ALA3633250 | 4 | pKi | = | 6.76 | ALA3636509 | 6.76 | nM | Homo sapiens | |||
| 20. | ALA3633250 | 4 | logD | = | -0.17 | ALA3636508 |
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