# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3634182 | 7A | Activity | 0 | ALA3635206 | Active | ||||||
2. | ALA3634182 | 7A | Activity | 0 | ALA3635205 | Active | ||||||
3. | ALA3634182 | 7A | EC50 | = | 0.04 | uM | ALA3635204 | 7.40 | nM | |||
4. | ALA3634182 | 7A | t1/2 | = | 15 | hr | ALA3635199 | hr | ||||
5. | ALA3634182 | 7A | t1/2 | = | 15 | hr | ALA3635198 | hr | Homo sapiens | |||
6. | ALA3634182 | 7A | Drug metabolism | = | 25.6 | % | ALA3635195 | % | Homo sapiens | |||
7. | ALA3634182 | 7A | Drug metabolism | = | 42 | % | ALA3635195 | % | Homo sapiens | |||
8. | ALA3634182 | 7A | Drug metabolism | = | 23.7 | % | ALA3635194 | % | Homo sapiens | |||
9. | ALA3634182 | 7A | Drug metabolism | = | 36.6 | % | ALA3635194 | % | Homo sapiens | |||
10. | ALA3634182 | 7A | INH | 0 | ALA3635193 | Not Active | % | |||||
11. | ALA3634182 | 7A | INH | = | 50 | % | ALA3635192 | % | ||||
12. | ALA3634182 | 7A | INH | 0 | ALA3635191 | Not Active | % | Rattus norvegicus | ||||
13. | ALA3634182 | 7A | IC50 | = | 0.6 | uM | ALA3635190 | 6.22 | nM | Rattus norvegicus | ||
14. | ALA3634182 | 7A | IC50 | = | 0.08 | uM | ALA3635190 | 7.10 | nM | Rattus norvegicus | ||
15. | ALA3634182 | 7A | INH | = | 50 | % | ALA3635187 | % | ||||
16. | ALA3634182 | 7A | IC50 | = | 12 | uM | ALA3635186 | 4.92 | nM | |||
17. | ALA3634182 | 7A | IC50 | = | 12.5 | uM | ALA3635186 | 4.90 | nM | |||
18. | ALA3634182 | 7A | Ratio IC50 | = | 2.5 | ALA3635185 | ||||||
19. | ALA3634182 | 7A | Ratio IC50 | = | 2.5 | ALA3635185 | ||||||
20. | ALA3634182 | 7A | EC50 | = | 0.003 | uM | ALA3637733 | 8.59 | nM | Homo sapiens |