| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA420540 | 22 | F | = | 15 | % | ALA637859 | % | ||||
| 2. | ALA420540 | 22 | AUC | = | 205 | ug min ml-1 | ALA638128 | ng.hr.mL-1 | ||||
| 3. | ALA420540 | 22 | AUC | = | 309 | ug min ml-1 | ALA638130 | ng.hr.mL-1 | ||||
| 4. | ALA420540 | 22 | T max | = | 90 | min | ALA638704 | hr | ||||
| 5. | ALA420540 | 22 | Cmax | = | 2.1 | ug ml-1 | ALA641863 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 6. | ALA420540 | 22 | T1/2 | = | 23 | min | ALA639886 | hr | ||||
| 7. | ALA420540 | 22 | T1/2 | = | 58 | min | ALA639888 | hr | ||||
| 8. | ALA420540 | 22 | Vdss | = | 230 | ml kg-1 | ALA638732 | L.kg-1 | ||||
| 9. | ALA420540 | 22 | Cl | = | 9.8 | ml min-1 kg-1 | ALA641609 | mL.min-1.kg-1 | ||||
| 10. | ALA420540 | 22 | F | = | 42 | % | ALA637852 | % | ||||
| 11. | ALA420540 | 22 | AUC | = | 457 | ug min ml-1 | ALA638129 | ng.hr.mL-1 | ||||
| 12. | ALA420540 | 22 | AUC | = | 363 | ug min ml-1 | ALA638131 | ng.hr.mL-1 | ||||
| 13. | ALA420540 | 22 | T max | = | 30 | min | ALA638704 | hr | ||||
| 14. | ALA420540 | 22 | Cmax | = | 3.8 | ug ml-1 | ALA641862 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 15. | ALA420540 | 22 | T1/2 | = | 54 | min | ALA639887 | hr | ||||
| 16. | ALA420540 | 22 | T1/2 | = | 68 | min | ALA639889 | hr | ||||
| 17. | ALA420540 | 22 | Vdss | = | 223 | ml kg-1 | ALA638733 | L.kg-1 | ||||
| 18. | ALA420540 | 22 | Cl | = | 5.9 | ml min-1 kg-1 | ALA875787 | mL.min-1.kg-1 | ||||
| 19. | ALA420540 | 22 | Selectivity | > | 10000 | ALA840708 | ||||||
| 20. | ALA420540 | 22 | Selectivity | > | 10000 | ALA840065 |
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